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2-({5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}(propan-2-yl)amino)ethan-1-ol
1-[(2-chlorophenyl)methyl]-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(5-phenoxyfuran-2-carbonyl)pyrrolidin-3-yl]methanol
3-(piperidin-1-ylmethyl)-1-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
(4aR,7aS)-1-cyclopropanecarbonyl-4-(3-fluoro-4-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(dimethylamino)-2-methylpropan-2-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-[2-(methylsulfanyl)benzoyl]piperidine
5-{3-[3-methyl-7-(2-methylpyrimidin-4-yl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]-1,2,4-oxadiazol-5-yl}pyrrolidin-2-one
(2S,4R)-4-{[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]amino}-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-{1-[(4-chloro-2-fluorophenyl)methyl]piperidin-3-yl}ethan-1-amine
7-(3-phenylpropyl)-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-[1-(1-benzylpiperidin-4-yl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]propanamide
[(3S,7S)-5-[4-(1H-imidazol-1-yl)benzoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
3-(2-ethylbutyl)-8-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-benzyl-2-(3-fluorophenyl)azepane-1-sulfonamide
2,2-dimethyl-3-[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]propan-1-ol
N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylbenzamide
methyl 4-[6-amino-5-cyano-4-(piperidin-4-yl)pyridin-2-yl]benzoate
3-(1-ethyl-1H-pyrazol-4-yl)-1-[3-(4-methylbenzenesulfonamido)propyl]urea
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(2-methoxyphenyl)propanamide
6-ethoxy-3-({[1-(methoxymethyl)cyclopropyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methylbenzamide
3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
4-{[5-(3-methyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-propylpiperidine
3-[(3R,4S)-1-(6-chloro-1,3-benzothiazol-2-yl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
5-(2,6-dimethoxyphenyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2,4-triazin-3-amine
4-fluoro-N-({1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-yl}methyl)benzamide
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-4-yl)-1,4-diazepan-6-ol
2-methanesulfonyl-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}acetamide
2-tert-butyl-8-cycloheptanecarbonyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(2-methanesulfonylethyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
{2-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazol-4-yl}methanol
1-(3-fluoro-2-methoxybenzoyl)-4-(3-methylpyridin-2-yl)piperazine
1-[(4-chlorophenyl)methyl]-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
1-[1-(1,7-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
2-amino-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,3-benzothiazole-5-carboxamide
ethyl 3-{[4-(carbamoylmethoxy)phenyl]formamido}propanoate
(1R,5S,8R)-3-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-8-methoxy-3-azabicyclo[3.2.1]octane
1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
3-ethyl-1-(1H-indol-5-ylmethyl)piperidine-3-carboxylic acid
5-methyl-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(3-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)cyclopentanamine
4-[4-(furan-2-carbonyl)piperazin-1-yl]-2-(thiomorpholin-4-ylmethyl)quinazoline
3-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)pyridine
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1H-indazole
4-methyl-2-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
(1R,3s,6r,8S)-4-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
2-chloro-N-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide