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methyl (2S)-3-carbamoyl-2-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}propanoate
1-methyl-3-(3-phenylpiperazine-1-carbonyl)-1,2-dihydropyridin-2-one
N-[(3S,4R)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1'-(2,4-dimethoxybenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-methoxy-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-(2-phenylacetyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
6-tert-butyl-1-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,5-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aR,8aR)-2-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-[(4-phenyloxan-4-yl)methyl]pyrrolidin-2-one
ethyl 2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetate
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
2-(2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[3-oxo-3-(pyrrolidin-1-yl)propyl]quinoxaline-5-carboxamide
1,6-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-benzyl-3-(2-methoxyethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-diethyl-2-({4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl}oxy)acetamide
(2R)-2-hydroxy-3-methyl-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-one
N-(1,4-dioxan-2-ylmethyl)-2-(4-fluorophenyl)-N-methylimidazo[1,2-a]pyridine-6-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}piperidin-2-one
N-(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
6-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
(1R,5R)-6-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-1,4-dihydropyridin-4-one
4-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}-1-[4-(propan-2-yl)phenyl]pyrrolidin-2-one
4-methyl-2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
2-{[(3-ethoxyphenyl)methyl]({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino}ethan-1-ol
1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-{4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-2-methylphenyl}pyridine-3-carboxamide
N-(2-methoxyethyl)-6-(4H-1,2,4-triazol-4-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyridine-3-carboxamide
4-(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)morpholine
4-(1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-3-yl)pyrimidine
2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-3-methylquinoxaline
2-{4-[(2-chloro-4,5-dimethoxyphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
ethyl 2-{4-[(thiomorpholine-4-carbonyl)amino]phenyl}acetate
3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-(propan-2-yl)-1,2-oxazole
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methylphenol
2-(1-benzothiophen-2-yl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-imidazole
N,N-dimethyl-2-[(1S,5R)-6-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]propanamide
2-cyclopropyl-8-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3S)-N-tert-butyl-2-(3-methyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-{2-[bis(propan-2-yl)amino]ethyl}-3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
N-[(3-methoxyphenyl)methyl]-3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]propanamide
N-[(4-hydroxyazepan-4-yl)methyl]-4-methyl-1H-imidazole-5-carboxamide
1-(carbamoylmethyl)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}piperidine-3-carboxamide
3-{[1-(oxolane-2-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
3-({[(3,4-difluorophenyl)methyl]amino}methyl)-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)propanamide