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4-[(5-ethylpyridin-2-yl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-one
N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(cyclopentylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclopropyl-3-[5-(2,5-dimethylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
methyl({[2-(propan-2-yl)pyrimidin-5-yl]methyl})[1-(pyridin-3-yl)ethyl]amine
2-methoxy-N-[6-methoxy-2-oxo-4-(quinolin-4-yl)-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
5-cyclobutyl-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
(2S,4R)-4-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
6-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
8-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-benzyl-11-({[3-(trifluoromethyl)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N5-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-methylphenyl)-5-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}-1,3-thiazole
1-[1-(furan-2-carbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
N'1-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]cyclopropane-1,1-dicarboxamide
1-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
4,6-dimethyl-2-oxo-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydropyridine-3-carboxamide
1-[(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-(1-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}piperidin-4-yl)methanesulfonamide
3-tert-butyl-1-methyl-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylfuran-2-carboxamide
2-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-[1-(3,4-dichlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
8-(5-chloro-3-fluoropyridin-2-yl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
3-[methyl({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amino]-1λ6-thiolane-1,1-dione
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-(3-cyclohexylpyrrolidin-1-yl)propan-1-one
7-(5-chloropyridin-2-yl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(methylsulfanyl)propan-1-one
[(2S,4R)-4-(dimethylamino)-1-[(5-methyl-1H-indol-3-yl)methyl]pyrrolidin-2-yl]methanol
3-methyl-N-propyl-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(furan-2-ylmethyl)piperidin-4-amine
1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)urea
7-[(4-fluorophenyl)methyl]-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-[3-(morpholin-4-yl)propyl]urea
N-[3-(1H-imidazol-2-yl)propyl]-3-(piperidin-3-yl)benzamide
2-{[4-(methylsulfamoyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)azetidin-3-ol
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
3,5-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1,2-oxazole-4-carboxamide
ethyl 2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]acetate
N-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)cyclopropanamine
1-(2-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-4,6-dimethylphenyl)-1H-pyrazole
3-(2-amino-1,3-thiazol-4-yl)-N-[(1R,2R)-2-(benzyloxy)cyclopentyl]propanamide
9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-2,7,8-trimethylquinoline
4-(3-methyl-1,2-benzoxazol-5-yl)-7-(2-oxo-1,3-oxazolidin-3-yl)-1,2,3,4-tetrahydroquinolin-2-one
N-[(4-chlorophenyl)methyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(2-oxopyrrolidin-1-yl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(3-ethoxy-4-methoxyphenyl)methyl]piperazine