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(2S)-N-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-2-(methoxymethyl)pyrrolidine-1-carboxamide
2-methyl-6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-[2-(2-chlorophenyl)ethyl]-4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridine-2-carboxamide
3-methyl-N-[(1R,2S)-2-phenylcyclopropyl]-1-propyl-1H-pyrazole-4-carboxamide
2-cyclopropyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyrimidine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-methylpiperidine
1-({1-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)azepane
5-[(1,3-benzothiazol-2-ylmethyl)amino]-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}quinoline
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[3-(1,3-oxazol-5-yl)phenyl]urea
4-{4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-(4-methyl-1H-imidazol-5-yl)-1-[(2,3,4-trimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-acetylphenoxy)-1-[7-(1-hydroxy-3-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
4-benzyl-3-ethyl-1-(pyridine-4-carbonyl)-1,4-diazepan-5-one
3-(4-cyclobutyl-6-methylpyrimidin-2-yl)-3,9-diazaspiro[5.6]dodecan-10-one
4-ethyl-3-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(methylsulfanyl)benzamide
2-[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]-6-methylpyridine-3-carboxylic acid
2-[1-(3-phenylpropyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-yl]ethan-1-ol
2-methoxy-N-{1-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
1-{4-[(5S,9aS,9bS)-1-oxo-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]phenyl}imidazolidin-2-one
4-(2-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)pyridine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[4-(2-oxopiperidin-1-yl)butanoyl]piperidine-3-carboxylate
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2H-indazol-2-yl)acetamide
N-(isoquinolin-5-ylmethyl)-N,2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(2-ethylbenzoyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-(cyclopropylamino)-N-{1-[(2-methylphenyl)methyl]cyclopropyl}acetamide
(1R,5S,8R)-8-(dimethylamino)-N-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide
5-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrazin-2-ol
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-methoxypyridine-4-carboxamide
7-{[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-2-ethyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
6-methyl-2-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}methyl)quinolin-4-ol
1-benzyl-3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrrolidine
6-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]pyridine-2-carboxylic acid
5-{[3-(trimethyl-1H-pyrazol-4-yl)propanamido]methyl}thiophene-2-carboxylic acid
3-fluoro-N-(1-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(2S)-1-{3-[(4-fluorophenyl)formamido]propanoyl}pyrrolidine-2-carboxamide
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-3-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-ethyl-2,5-dimethyl-1H-pyrrole-3-carboxamide
N-ethyl-N-(4-hydroxybutyl)-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
(1S,5R)-3-[4-(pyridin-4-yl)pyrimidin-2-yl]-3,9-diazabicyclo[3.3.2]decan-10-one
8-(9H-fluoren-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
3-[(4aR,7aS)-4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-(4-tert-butylbenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
2-{2-[4-phenyl-1-(thiolan-3-yl)-1H-imidazol-5-yl]-1H-pyrrol-1-yl}pyrimidine
4-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-5-phenyl-1,2-oxazole
N,N-dimethyl-2-(2-phenylpyrimidin-5-yl)quinoline-4-carboxamide