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2-[N-(4-methylphenyl)methanesulfonamido]-N-[3-(pyridin-4-yl)propyl]acetamide
2-ethyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
N-[(2S,4R,6R)-2-(2-butyl-1H-imidazol-4-yl)-6-(4-chlorophenyl)oxan-4-yl]acetamide
1-methyl-6-propyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(4-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)pyrazine-2-carbonitrile
[1-(4-methylpyridin-2-yl)-1H-1,3-benzodiazol-2-yl]methanol
4-methyl-5-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
(3S,9aR)-3-benzyl-8-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(furan-2-ylmethyl)-3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
5-ethyl-N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-methylpyrimidin-4-amine
2-(8-methoxy-2-methylquinolin-5-yl)pyridine-4-carboxamide
2-(methylsulfanyl)-5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyrimidine
(5-{[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]methyl}furan-2-yl)methanol
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(3-phenoxyphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
3-methyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-dihydroquinoxalin-2-one
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-4-oxo-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl]urea
N-cyclopropyl-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
2,6-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]quinoline-3-carboxamide
2-methyl-6-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-benzoxazole
1-[(2S,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
2-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
[(2S,6S)-4-{[4-(trifluoromethyl)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-N-(2-phenylethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2-[(2,4-dimethoxyphenyl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
(2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,4-diazepan-2-one
8-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)quinoline
7,11-dimethyl-3-[4-(pyridin-3-yl)pyrimidin-2-yl]-3,7,11-triazaspiro[5.6]dodecane
methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
4-[(4-methoxyphenyl)methyl]-1-(5-methyl-1H-indole-2-carbonyl)-1,4-diazepan-5-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(thiophen-2-yl)ethyl]urea
N-[(3S,5S)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-4-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-6-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-6-azaspiro[2.5]octane-1-carboxamide
[(1-{[1-(2-phenylpropyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]urea
2-({2-[({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)carbamoyl]phenyl}amino)acetic acid
5-[({[2-(butan-2-yl)phenyl]carbamoyl}amino)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(3-methylpyrazin-2-yl)-decahydro-1,6-naphthyridin-2-one
2-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(1-benzyl-1H-pyrazole-4-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
8-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(1R,9aR)-1-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}-octahydro-1H-quinolizin-1-ol
N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]oxane-4-carboxamide