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5-[(dimethylamino)methyl]-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,3,4-oxadiazole-2-carboxamide
3-{[5-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
(3aS,6aS)-2-(cyclopropylmethyl)-5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-propyl-2-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
1-(furan-2-ylmethyl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]piperidine-4-carboxamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-(1H-indol-3-yl)acetamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-(1-benzothiophen-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-4-methyl-1H-imidazole-2-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
8-[(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(isoquinolin-5-ylmethyl)-1-(2-methoxyethyl)-N-methyl-6-oxopiperidine-3-carboxamide
4-{[2-(adamantan-1-yl)-4-hydroxypyrimidin-5-yl]formamido}-N-methylbutanamide
4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N,N-dimethylpiperazine-1-sulfonamide
3-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
N-[2-(3-phenoxyphenyl)ethyl]pyrrolidine-3-carboxamide
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N,4,6-trimethyl-2-oxo-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1,2-dihydropyridine-3-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-(2-methyl-1,3-benzoxazole-6-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
1-{2-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexane-3-carbonyl]phenyl}-1,3-diazinane-2,4-dione
(1-benzothiophen-2-ylmethyl)({[6,7-dimethoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
3-(2-hydroxyethyl)-4-(2-methyl-1-benzofuran-7-carbonyl)piperazin-2-one
benzyl N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
4-({[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}(methyl)amino)-1λ6-thiane-1,1-dione
1-(2-chlorophenyl)-4-[2-(1H-pyrazol-1-yl)butanoyl]piperazin-2-one
3-(3-methoxyphenyl)-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
(3S,9aR)-8-(cyclopropylmethyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-chlorobenzoic acid
N-(oxan-4-yl)-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
5-({4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}methyl)-2-methoxybenzoic acid
5-methyl-1-phenyl-4-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperazin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(3S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-(3-methoxypropyl)-1-methyl-N-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-amine
3-[4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
[(1-methylpiperidin-4-yl)methyl](2-phenylethyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
3-(2-methylpropyl)-2-oxo-1-(prop-2-en-1-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
1-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4-(pyridin-4-yl)piperazine
N-methyl-N-{2-phenyl-1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]ethyl}thiophene-2-carboxamide
N-ethyl-2-(ethylamino)-N-[2-(4-fluorophenoxy)ethyl]pyrimidine-5-carboxamide
N-cyclopropyl-1-[1-(quinolin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
1-[(3-chloro-4-hydroxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N-[2-(dimethylamino)ethyl]-5-[1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-{1-[(2-chloro-4,5-dimethoxyphenyl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methanesulfonylpiperidine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-3-(methylsulfanyl)-N-(oxolan-2-ylmethyl)propanamide
1-(4-{2-oxo-2-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)propan-1-one