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2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-propylacetamide
N-(1H-indazol-7-yl)-2-(pyrrolidin-3-yl)benzamide
1-{2-[1-(isoquinolin-5-ylmethyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-methoxybenzamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[2-(methylsulfanyl)benzoyl]pyrrolidin-3-amine
N-(2-oxopiperidin-3-yl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
1-[1'-(2,5-dimethylfuran-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N,N-diethyl-1-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-6-(pyrrolidin-1-yl)pyrimidine
2-amino-8-[4-ethoxy-3-(hydroxymethyl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(2S,4S)-4-amino-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(5-methylfuran-2-yl)phenyl]-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
2-[4-carbamoyl-4-(piperidin-1-yl)piperidin-1-yl]-2-(2-fluoro-4-methylphenyl)acetic acid
5-[methyl(prop-2-yn-1-yl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-2-(1H-pyrazol-1-yl)benzamide
N-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]quinoline-8-sulfonamide
N-methyl-N-(2-phenylethyl)-5-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-methyl-7-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
8-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
7-(quinolin-3-yl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
N-[2-(4-phenylpiperidin-1-yl)ethyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[4-(dimethylamino)phenyl]acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
[1-(1-benzothiophen-2-ylmethyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
3-({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylpropanamide
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-(piperidin-3-ylmethyl)pyrimidine-5-carboxamide
3-(2-methylphenyl)-3-phenyl-N-[(1r,4r)-4-hydroxycyclohexyl]propanamide
methyl 2-{4-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
2-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}-1-(propan-2-yl)-1H-1,3-benzodiazole
1-(2-methoxyphenyl)-5-methyl-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperazin-2-one
1-[3-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-3-oxopropyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyphenoxy)acetamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N,1-dimethyl-N-[3-(1H-pyrazol-1-yl)propyl]pyrrolidine-3-carboxamide
4-(cyclopropylmethyl)-1-[3-(hydroxymethyl)-7-methylquinolin-2-yl]piperidine-4-carboxylic acid
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
1-(4-chloro-1H-indole-2-carbonyl)azetidin-3-ol
N-(cyclopropylmethyl)-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-1,3-oxazole-4-carboxamide
2-[4-(9H-purin-6-yl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
2-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)formamido]acetamide
5-{[methyl({[3-(2-{4-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(2-hydroxybenzoyl)piperidine-3-carboxylic acid
1-[(2-methoxyphenyl)methyl]-6-oxo-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide