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({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)(pentan-3-yl)amine
4-(2-methyl-1H-imidazol-1-yl)-1-(quinolin-2-yl)piperidine-4-carboxylic acid
2-[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
N-(4-{[(5-oxo-1-propylpyrrolidin-3-yl)carbamoyl]methyl}phenyl)butanamide
5-methyl-N-(2-phenylethyl)-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
1-(2-methylphenyl)-4-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]piperazin-2-one
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(2-methyl-1H-imidazol-1-yl)acetamide
5-(5-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)-1H-1,3-benzodiazole
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(3-methyl-1-benzothiophene-2-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(oxan-2-ylmethoxy)ethan-1-one
{[1-(1-hexylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}(methyl)amine
2-[1-(3,3,3-trifluoro-2-methylpropyl)azetidin-3-yl]-1H-1,3-benzodiazole
2-(4-fluorophenyl)-1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
3-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
4-benzyl-3-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-(1,4-dioxan-2-ylmethyl)-N-methylpyridin-2-amine
4-{butyl[2-(1-methylpiperidin-2-yl)ethyl]amino}butan-1-ol
2-methoxy-6-({[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)amino}methyl)phenol
N1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}propane-1,3-diamine
2,2-dimethyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}butanamide
3-({5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}methyl)-5-ethyl-1,2,4-oxadiazole
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]piperazine
2-{[(1S,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amine
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
4-fluoro-N-({1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}methyl)benzamide
N-[(3R,4S)-4-(propan-2-yl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-yl]methanesulfonamide
1-[2-(pyridin-3-yl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
3-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-3-yl]benzoic acid
3-[(propan-2-yl)sulfamoyl]-5-(1H-pyrazol-4-yl)benzoic acid
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
N-(2-acetamidoethyl)-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-[2-(3-methylthiophen-2-yl)ethyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
1-[4-(hydroxymethyl)benzoyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
3-{[1-(hydroxymethyl)cyclopropyl]methyl}-3-methyl-1-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
1-methyl-4-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[2-(6-hydroxypyrimidin-4-yl)ethyl]-5,5-diphenylpiperidin-2-one
N-methyl-2-oxo-N-phenyl-2-(3-propoxypiperidin-1-yl)acetamide
5-{2-[(2-phenoxyethyl)amino]ethyl}-1-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
2-(4-benzoyl-6-hydroxy-1,4-diazepan-1-yl)pyridine-4-carbonitrile
3-{5-[2-(pyridin-4-ylsulfanyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
(2R,6R)-4-[4-(hydroxymethyl)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-methylazepane-2-carboxamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-[3-({[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
1-(4-fluorophenyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,4-diazepane
1-(3-hydroxyphenyl)-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide