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3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-[2-(dimethylamino)ethyl]pyrrolidin-2-one
3-(2-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-2-oxoethyl)-4,6-dimethyl-2,3-dihydro-1H-indol-2-one
1-[(1-ethylpyrrolidin-3-yl)methyl]-1,2-dihydroquinolin-2-one
N-[(1-cyclopentylpyrrolidin-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-benzoyl-N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-amine
2-[1-(thiophen-2-yl)ethyl]-4-(4-{[4-(trifluoromethoxy)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N-(pyridin-3-ylmethyl)-4-(quinolin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{3-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
(3R,4R)-4-cyclobutyl-3-methyl-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-ol
5-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-indole-2-carboxamide
6-fluoro-2-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}quinolin-4-ol
5-cyclopropyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(3R,4R)-1-(2-amino-9H-purin-6-yl)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
8-(1-methoxypropan-2-yl)-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
2-methanesulfonyl-6-methyl-5-[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
4-{6-[2-(1,3-thiazol-2-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
2-(2-methyl-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-(3-{4-[(pyridin-3-ylmethyl)amino]piperidin-1-yl}phenyl)cyclopropanecarboxamide
N-(2-methylprop-2-en-1-yl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)propanamide
3-(5-methylfuran-2-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
6-(4-chlorophenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[1-(quinoxaline-6-carbonyl)piperidin-3-yl]benzoic acid
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(2,5-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,7,8-trimethyl-4-(3-methylpiperidine-1-carbonyl)quinoline
N-(4-{[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]methyl}phenyl)acetamide
4-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-1,4-oxazepan-6-ol
2-[(5-cyclopentylthiophen-2-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-{1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-imidazol-2-yl}benzonitrile
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)cyclopropanamine
(2,1,3-benzoxadiazol-4-ylmethyl)[(1-ethylpyrrolidin-2-yl)methyl]{[1-(2-methoxyethyl)piperidin-4-yl]methyl}amine
1-[(4-methoxyphenyl)methyl]-N-methyl-N-(pyrazin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[4-(5-fluoro-2-methoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
methyl(2-{4-methyl-2-[3-(1H-pyrazol-3-yl)phenyl]phenoxy}ethyl)amine
4-(benzyloxy)-1-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
6-amino-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]hexan-1-one
methyl 2-(diethylsulfamoyl)-6-(3-fluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-1-cyclopentylpiperazin-2-one
1-cyclopropyl-4-{4-[(4-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrrolidin-2-one
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-(piperidin-4-yl)pyridin-2-amine
3-{2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-4-(2-methylpropyl)piperazin-2-one
N-[(1S,6R)-6-carbamoylcyclohex-3-en-1-yl]-N'-(4-methylphenyl)propanediamide
4-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]thiomorpholine
4-[2-(4-phenyl-5-propyl-1H-imidazol-1-yl)ethyl]pyridine
2,6-dimethoxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyridine-3-carboxamide