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methyl 2-(5-methyl-2-{[(3-methylfuran-2-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
N-[3-(cyclohexyloxy)propyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
8-methyl-5-{1-[1-(pyrimidin-4-yl)ethyl]-1H-imidazol-2-yl}quinoline
7-[(3,4-difluorophenyl)methyl]-2-(2-methylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-{1-[(thiophen-2-ylmethyl)carbamoyl]piperidin-3-yl}benzoic acid
2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoline
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-(5-methyl-1H-pyrazol-1-yl)acetamide
4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-3-(3-fluorophenyl)piperazin-2-one
N-(propan-2-yl)-6-(3,4,5-trimethoxyphenyl)pyrimidin-4-amine
1-methyl-4-[5-(pyrrolidin-1-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]-1,4-diazepane
4-benzyl-7-(2,3-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
4-(5-methoxypyridin-3-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(2-{1-[(5-chloro-1,3-benzoxazol-2-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
7-(cyclopropylmethyl)-2-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
5-(4-acetyl-2-methoxyphenoxymethyl)-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide
5-ethyl-N-({7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,2-oxazole-3-carboxamide
5-tert-butyl-4-({7,9-dioxo-8-azaspiro[4.5]decan-8-yl}methyl)furan-2-carboxamide
2-methyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2,3-dihydropyridazin-3-one
1-[(2,3-difluorophenyl)methyl]-3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-3-phenyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyridine-3-carboxamide
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]cyclobutanecarboxamide
2-[4-(4-{[2-(1H-imidazol-4-yl)ethyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-yl]phenol
methyl 1-(2-methoxyethyl)-3-(3-phenylpropanamido)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-N-[(3-methylthiophen-2-yl)methyl]cyclopentanamine
2-{[(4-fluorophenyl)methyl](quinoxalin-2-ylmethyl)amino}butan-1-ol
N-methyl-5-(1-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
ethyl 1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine-4-carboxylate
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N,5-dimethyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
N-(1-methyl-1H-pyrazol-5-yl)-4-({methyl[1-(pyridin-3-yl)propyl]amino}methyl)benzamide
1-[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[(3-fluorophenyl)methyl]-N-[2-(4-methylphenyl)ethyl]-6-oxopiperidine-3-carboxamide
4-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
7-[1-(4-fluorophenyl)cyclopropanecarbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidine-1-sulfonyl)piperazine
6-cyano-N-{[2-(diethylamino)pyridin-3-yl]methyl}pyridine-3-carboxamide
(3S,4R)-4-phenyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-3-carboxylic acid
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)spiro[2.2]pentane-1-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]ethan-1-one
9-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
1-(4,6-dimethylquinazolin-2-yl)-N-(1,4-dioxan-2-ylmethyl)piperidine-4-carboxamide
(1S,5R)-6-propyl-3-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(2-chlorophenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]furan-2-carboxamide
7-{[4-(propan-2-yl)phenyl]methyl}-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
4-(dimethylamino)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
3-{[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]sulfamoyl}-N-propylbenzamide
(1S)-1-[1-(2,5-dichlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethan-1-amine