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3-cyclopropyl-5-(4-phenylbutyl)-1H-1,2,4-triazole
4,6-dimethyl-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(1H-imidazol-2-ylmethyl)piperidine-4-carboxylic acid
ethyl 2-[1-(2,3-dimethoxybenzoyl)piperidin-2-yl]acetate
2-{4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}pyridine-3-carboxamide
N,1-dimethyl-6-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(3-chloro-4-hydroxybenzoyl)-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
2-[4-(4-ethylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
N4-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidine-2,4-diamine
1-(2,3-dihydro-1H-inden-5-yl)-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-methylurea
1-methyl-2-[5-(5-methylpyrazin-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-1H-1,3-benzodiazole
{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
4-(cyclohexylamino)-1-(2,2-dimethylpropyl)pyrrolidin-2-one
1-(oxolane-3-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methoxyhexan-1-one
N-cyclopropyl-5-[2-(1H-indazol-3-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-(2-methylpyrimidin-4-yl)piperidin-3-yl]propan-1-ol
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(4-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
N,N-dimethyl-2-(4-{6-[(thiophen-2-ylmethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperazin-1-yl)acetamide
6-ethyl-N-[4-(furan-2-yl)butan-2-yl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]pyridine-3-carbonitrile
1,3-dimethyl-4-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperazin-2-one
3-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
4-(piperidine-1-carbonyl)-1-(1H-pyrrole-3-carbonyl)piperidine
N3-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
(5R)-5-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyrrolidin-2-one
3-({methyl[(1-phenylpyrrolidin-3-yl)methyl]amino}methyl)phenol
3-[(4-ethylpiperazin-1-yl)methyl]-1-(prop-2-en-1-yl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
2-[4-(methylsulfanyl)phenyl]-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
1-ethyl-3-methyl-4-[(E)-2-phenylethenyl]-1H-pyrazole
2-[(4-benzylpiperazin-1-yl)methyl]-N-(furan-3-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
(3S,5S)-5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1-methylpyrrolidin-3-amine
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-[2-(pyrrolidin-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-aminoethyl)-N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methylquinazolin-4-amine
(4aS,7aR)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-ethyl-3-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N,5,7-trimethyl-N-(oxan-2-ylmethyl)pyrido[2,3-d]pyrimidin-4-amine
1-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperidine-4-carboxamide
4-(2-methyl-1-benzofuran-7-carbonyl)thiomorpholine
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(3-methoxypropyl)-N-methylpiperidine-3-carboxamide
7-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
4-(piperidin-1-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]butanamide
2-fluoro-5-[2-(4-fluorophenoxy)ethyl]benzamide
4-fluoro-N-({1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]piperidin-3-yl}methyl)benzamide
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
6-fluoro-2-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}quinolin-4-ol
1-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-5-oxopyrrolidine-3-carboxylic acid
propyl 4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate