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N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2S,4S)-4-amino-1-[4-(4-fluorophenyl)oxane-4-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(pyrazin-2-yl)-2-({2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)acetamide
4-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]-1,4-oxazepan-6-ol
methyl 5-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-methylazepan-4-ol
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(2-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[3-(1H-pyrazol-1-yl)benzoyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
2-{[4-(2-chlorophenyl)-5-[hydroxy(phenyl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-4-methylbenzamide
1-(2,6-dimethylphenyl)-3-{2-[(2R)-pyrrolidin-2-yl]ethyl}urea
5-fluoro-2-[1-(furan-2-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
N-[(8-methoxyquinolin-5-yl)methyl]-N,6-dimethyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-methoxy-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1,2-dihydropyridin-2-one
methyl({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1,5-dimethyl-4-({2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
7-chloro-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
2-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)pyridine-3-carboxylic acid
1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-[(4-fluorophenyl)methyl]piperidine
1-(cyclohexylmethyl)-3-hydroxy-3-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)piperidin-2-one
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1,9-dioxaspiro[5.5]undecan-4-amine
methyl 6-{[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)carbamoyl]amino}-1,2,3,4-tetrahydroquinoline-1-carboxylate
3-methoxy-2,2-dimethyl-N-[(1R,2S)-2-phenylcyclopropyl]propanamide
(1S,5R)-3-methyl-6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
2-(4-chlorophenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-methyl-3-(2-phenylethyl)-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
8-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{3-[(4-methoxyphenyl)methyl]-1-methyl-1H-1,2,4-triazol-5-yl}-2-methylpyridine
2-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine-4-carbonitrile
(1R,5R)-6-(cyclobutylmethyl)-3-(3-phenyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(1H-imidazol-2-ylmethyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
4-methoxy-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-[(2-methoxynaphthalen-1-yl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(1-cycloheptylpiperidin-3-yl)methyl]-1,3-thiazole-5-carboxamide
1-[1-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
(2S,4R)-4-amino-N,N-diethyl-1-(pyrimidin-2-yl)pyrrolidine-2-carboxamide
8-{[3-(morpholin-4-ylmethyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-3,5,7-trimethyl-1H-indole
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
2-ethyl-N-{[1-(pyridin-3-ylmethyl)piperidin-3-yl]methyl}pyrimidine-5-carboxamide
2,4-dimethoxy-5-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]pyrimidine
1-ethyl-5-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methoxypiperidine
methyl 8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[(3R,4S)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)amino]-4-propylpyrrolidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
4-[(2-chlorophenyl)methyl]-1-[2-(methylsulfanyl)benzoyl]-1,4-diazepan-5-one