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3-(1H-1,2,3-benzotriazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
4-fluoro-N-{3-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}benzamide
3-phenyl-1-[1-(quinoline-5-carbonyl)piperidin-4-yl]propan-1-ol
1-{4-[(4-methoxypiperidin-1-yl)methyl]thiophen-2-yl}ethan-1-one
N-[(1S,2R)-2-aminocyclobutyl]-3-(2-methoxyphenyl)benzamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pent-4-enoyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2-methoxyphenyl)methyl]-2-{[(3S)-2-oxoazepan-3-yl]amino}acetamide
5-methyl-4-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)-2-[4-(methylsulfanyl)phenyl]-1,3-oxazole
1-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
[2-(azepan-1-yl)ethyl](ethyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-(4-cyano-2,5-difluorophenyl)-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea
(3R)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N,N-diethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]aniline
methyl (2S,4R)-1-[4-(4-chlorophenoxy)piperidine-4-carbonyl]-4-hydroxypyrrolidine-2-carboxylate
4,5-dimethyl-6-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}pyrimidine
1-[2-(4-methoxyphenyl)ethyl]-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[9-(4-hydroxy-3-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
2-(2-aminoethyl)-N-(5-methylpyridin-3-yl)morpholine-4-carboxamide
methyl 1-methyl-2-(1H-pyrazol-3-yl)-1H-1,3-benzodiazole-5-carboxylate
1-[(4-methylphenyl)methyl]-5-oxo-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]pyrrolidine-3-carboxamide
methyl (2S)-1-[3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 3-(2-chlorobenzenesulfonamido)-5-{[(3-methoxyphenyl)formamido]methyl}benzoate
N-({3-methyl-7-[2-(morpholin-4-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
(2S,4R)-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
5-[2-(1H-pyrazol-4-yl)ethyl]-3-(thiophen-3-yl)-1,2,4-oxadiazole
N-(2-chlorophenyl)-3-[1-(pyrrolidine-1-sulfonyl)piperidin-4-yl]propanamide
1-(1H-pyrrole-2-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})(pyridin-4-ylmethyl)amine
N-butyl-2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-1H-1,2,4-triazole-5-carboxamide
6-{methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-N'-(4-methoxyphenyl)propanediamide
9-[(3,5-dimethoxyphenyl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-propoxypiperidine
(2S)-2-amino-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}pentanamide
(3R)-3-methyl-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
(3S,4R)-1-(2-methoxyacetyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-[(3-fluorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
2-(3-methoxybenzamido)-7-oxo-N-[(3S)-2-oxoazepan-3-yl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-[2-(dimethylamino)ethyl]-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
7-(3-hydroxypyridine-2-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(3-fluoro-4-methylphenyl)-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-{[1-(3-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methoxy}acetamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
4-[(dimethylamino)methyl]-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}azepan-4-ol