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methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-ethoxypropan-1-one
(3R)-1-{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}pyrrolidin-3-ol
[3-(cyclopropylmethyl)-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]methanol
1-[(2-chlorophenyl)methyl]-4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazole
2-[1-({1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-6-methoxy-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-methyl-8-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-(2-methyl-1H-imidazol-1-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-(4-fluorophenyl)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-4-ol
N-(1-benzylpyrrolidin-3-yl)-5-methyl-4-{[(5-methylfuran-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
3-[(4-pentyl-1H-1,2,3-triazol-1-yl)methyl]-1λ6-thiolane-1,1-dione
4-methoxy-N-(2-methoxyethyl)-2-({1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}oxy)benzamide
3-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-{2-[(3-methylpyridin-4-yl)amino]ethyl}urea
methyl 2-({[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)amino)acetate
7-(cyclohexylmethyl)-2-(6-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
7-(1,2-oxazole-3-carbonyl)-N-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-benzoyl-2-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidine
2-amino-7-(2-amino-3-cyclopentylpropanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
{4-[(3-fluorophenyl)methyl]-1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}methanol
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N,2,8-trimethylquinoline-4-carboxamide
2-ethyl-4-[(2E)-3-phenylprop-2-en-1-yl]-1-(propan-2-yl)piperazine
7-chloro-N-[2-(furan-2-yl)ethyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
2-(2-methylpyridin-4-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
6-[(dimethylamino)methyl]-N-[4-(pyridin-3-yloxy)phenyl]-1,4-oxazepane-4-carboxamide
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-3-(1-methylpiperidin-2-yl)propanamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-(4-methoxyphenyl)pyrimidine
2-{4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
5-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
1-(furan-3-carbonyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepan-6-ol
4-(4-benzamidopiperidin-1-yl)pyrimidine-5-carboxylic acid
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-ol
1'-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{4-cyclohexyl-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(2,3-dihydro-1H-inden-1-yl)acetamide
4-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-4-oxobutane-1-sulfonamide
ethyl 1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylate
N-cyclopropyl-3-[5-(oxolan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
4-{[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]methyl}benzoic acid
2-(3,5-dimethyl-1-benzofuran-2-yl)-1-(2-methanesulfonylethyl)-1H-imidazole
2-benzyl-8-(cyclopropanesulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-6-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-1H-indole
4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-(2-methoxyphenyl)piperazin-2-one
ethyl 3-benzyl-1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidine-3-carboxylate
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
(4aS,8aR)-6-[2-(1H-imidazol-1-yl)acetyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine