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1-(dimethyl-1,2-oxazole-4-carbonyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chloro-4-fluoro-1-benzothiophene-2-carboxamide
5-(1H-indol-6-yl)-1,2,3,4-tetrahydroisoquinoline
2-(2,5-dimethoxyphenyl)-1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2-{methyl[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)cyclopentan-1-ol
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
1-[4-(4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)phenyl]ethan-1-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)ethan-1-one
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]pyrrolidine-2-carboxamide
1-[4-(3-benzyl-4H-1,2,4-triazol-4-yl)phenyl]ethan-1-one
(3R,5R)-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
4-[(1-benzothiophen-2-ylmethyl)amino]-5-methyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
[1-(1,3-benzothiazol-2-ylmethyl)-4-[(2-chlorophenyl)methyl]piperidin-4-yl]methanol
[(3R,4R)-1-(5-chloropyridin-2-yl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(2-methoxyphenyl)-2-methylpiperazine
8-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
2-[2-(4-fluorophenyl)morpholin-4-yl]-N-(propan-2-yl)pyridine-4-carboxamide
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
1-(4-{[2-(diethylamino)ethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
9-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,4,9-triazaspiro[5.5]undecan-5-one
1-[3-(5-methylfuran-2-yl)butyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-(2-hydroxyphenoxy)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]acetamide
methyl 2-{[5-(4-fluorophenyl)-4-[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
3-(methanesulfonylmethyl)-5-(1-phenylcyclopentyl)-1,2,4-oxadiazole
(2S,4R)-4-(2,4-dimethoxybenzamido)-N-ethyl-1-propanoylpyrrolidine-2-carboxamide
4-[2-(1-methyl-1H-pyrazol-4-yl)phenoxy]thiane-4-carboxylic acid
(2E)-N-tert-butyl-3-phenyl-N-(pyridin-2-ylmethyl)prop-2-enamide
5-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-oxazol-3-ol
2-cyclopropyl-N-{2-[ethyl(3-methylphenyl)amino]ethyl}-4-hydroxypyrimidine-5-carboxamide
methyl 2-({3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}amino)benzoate
N-(oxolan-2-ylmethyl)-4-({[2-(pyrazin-2-yl)ethyl]carbamoyl}amino)benzamide
N3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
4-{[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
methyl 4-[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})carbamoyl]benzoate
N-{5-[3-(1H-pyrazol-3-yl)phenyl]pyridin-2-yl}butanamide
3-phenyl-1-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]propan-1-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[3-(pyridin-2-yl)propyl]acetamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-[4-chloro-2-({[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)phenoxy]acetamide
N-methyl-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
2-methyl-3-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-indole
(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
[(5-chlorofuran-2-yl)methyl][(5-cyclopropyl-1,2-oxazol-3-yl)methyl]methylamine
2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3,3,3-trifluoro-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one