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N-methyl-N-[2-(oxan-4-yl)ethyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-{3-[2-chloro-5-(trifluoromethoxy)phenyl]-1-methyl-1H-1,2,4-triazol-5-yl}morpholine
6-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
{1-[6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}(thiophen-2-yl)methanol
4-(hydroxymethyl)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}azepan-4-ol
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
8-(2-hydroxybenzoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-oxo-8-(5-propyl-1,3,4-thiadiazol-2-yl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(3-methoxyphenyl)-3-[1-(pyridine-3-sulfonyl)piperidin-4-yl]propanamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-4-acetamidobenzamide
methyl 1-(2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperidine-4-carboxylate
N-{2-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}methanesulfonamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}propanamide
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
5-(2,6-difluoro-3-methylphenyl)-1-(1,4-dioxan-2-ylmethyl)-4-phenyl-1H-imidazole
1-{1-[4-(propan-2-yloxy)benzoyl]piperidin-4-yl}piperidin-3-ol
2-methyl-4-oxo-N-[(1R)-1-phenylpropyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
(1R,2S)-N-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-2-phenylcyclohexan-1-amine
1-(2-methoxyethyl)-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
2-[4-(3-methylphenoxy)piperidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,4-diazepan-5-one
N-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
3-[(1-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}propan-2-yl)oxy]pyridine
3-(oxan-2-ylmethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
5-(1-{[1-(methoxymethyl)cyclopropyl]methyl}-4-phenyl-1H-imidazol-5-yl)isoquinoline
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
(1R,5S)-3-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3,8-diazabicyclo[3.2.1]octane
1-benzyl-8-(9H-fluoren-2-ylmethyl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[(3,4-dimethoxyphenyl)formamido]ethyl}-N-phenyl-1H-1,2,3-triazole-4-carboxamide
3-{1-[(2-aminopyrimidin-5-yl)methyl]piperidin-4-yl}-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-ethyl-3-(oxan-2-ylmethyl)-1-[4-(pyridin-3-yloxy)phenyl]urea
2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-6-fluorobenzonitrile
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
4-(2,5-dimethoxyphenyl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)phenol
6-(2-chlorophenyl)-N-(2-methoxyethyl)-N-(propan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}-3-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione
N-[1-(thiophene-2-carbonyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
methyl (2S)-1-({4-[(2-butyl-1H-imidazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
3-hydroxy-1-[(3-methylphenyl)methyl]-3-{[(2-phenylpropan-2-yl)amino]methyl}piperidin-2-one
1-(2-methoxy-6-{[(2-phenoxyethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-(4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)-6-methylpyridazine
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
(2S,4S)-1-(2,2-diphenylethyl)-4-{[(2-fluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
ethyl 1-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine-3-carboxylate
4-(2-amino-6-methylpyrimidin-4-yl)-N,N-diethylbenzamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-(3-chloro-4-hydroxyphenyl)ethan-1-one
5-chloro-2-methoxy-4-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]pyridine
3-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one