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(2R)-2-amino-4-methyl-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}pentanamide
[(2S)-1-(4-{[(3-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidin-2-yl]methanol
N-(propan-2-yl)-1-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
methyl 5-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-(4-methoxyphenyl)-4-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]piperazine
5-{2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{1-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperidin-4-yl}phenol
N-[4-({[1-(4-ethoxyphenyl)ethyl]carbamoyl}methyl)phenyl]butanamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-methoxypropan-1-one
3-methoxy-6-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]pyridazine
N-[5-(2-fluoro-6-methoxyphenyl)-6-methylpyridin-2-yl]propanamide
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrimidine
2-{5-[(2S)-1-(1H-1,2,4-triazole-5-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(isoquinoline-5-carbonyl)pyrrolidin-3-yl]methanol
N-[3-(dimethylcarbamoyl)-5-({[1-(4-hydroxy-3-methoxyphenyl)propan-2-yl]amino}methyl)phenyl]pyridine-2-carboxamide
(2-ethoxy-5-{[methyl(oxan-2-ylmethyl)amino]methyl}phenyl)methanol
3-(2,3-dihydro-1H-indol-1-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
(2S,4R)-N-ethyl-1-(pyridin-4-ylmethyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(3aR,6aS)-5-(6-cyanopyridine-3-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-(1H-indole-6-carbonyl)-N-[4-(1H-pyrazol-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
[(4-ethoxyphenyl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
3-({[1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
(3S,4S)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-(quinolin-4-yl)pyrrolidin-3-ol
5-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-(methylsulfanyl)pyrimidine
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-benzyl-8-(2-methoxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
(1S,4S)-2-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-2-azabicyclo[2.2.1]heptane
3-(2-hydroxyethyl)-4-(5-methyl-2-phenylfuran-3-carbonyl)piperazin-2-one
2-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}-2,7-diazaspiro[4.5]decan-6-one
7-(2-phenylethyl)-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
3-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}phenol
6-(2,5-dimethylfuran-3-yl)-N-[(5-methylfuran-2-yl)methyl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-methoxy-1-{1'-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
3-[(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
1,3-dimethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(2-{[1-(6-chloro-2-methylquinoline-4-carbonyl)piperidin-4-yl]oxy}ethyl)dimethylamine
1-[(4-chlorophenyl)methyl]-N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(3S,5S)-5-(morpholine-4-carbonyl)-1-[(2-propylpyrimidin-5-yl)methyl]piperidine-3-carboxylic acid
1-[4-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)phenyl]pyrrolidin-2-one
2-{1-cyclohexyl-4-[(4-ethynylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4,6-dimethyl-3-{4-[(pyrimidin-2-yl)amino]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-[4-(6-aminopyrimidin-4-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
(4-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}morpholin-2-yl)methanamine
2-({[(3R,4R)-1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[benzyl(methyl)amino]-3-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]propan-2-ol
4-[3-(2-methoxyethyl)-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-phenylethan-1-one
(1S,2R)-N2-tert-butyl-N1-(2-methoxyethyl)-N1-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclohexane-1,2-dicarboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one