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(2R)-2-[(1-benzyl-4-phenylpiperidin-4-yl)formamido]propanoic acid
2-{4-[(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)methyl]-3,5-dimethyl-1H-pyrazol-1-yl}ethan-1-ol
N-[(3S,5S)-1-cyclopentyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-phenyl-N-[2-(pyridin-3-yloxy)propyl]imidazo[1,2-a]pyridine-6-carboxamide
2-[2-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
3-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-6-chloro-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
(2R,3R)-3-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(5-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
{2-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]ethyl}dimethylamine
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(quinolin-2-ylmethyl)piperidine-2-carboxamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
1-(2-{methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
(1S,5R)-6-benzyl-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-[1-(3-hydroxy-4-methoxybenzoyl)piperidin-3-yl]piperazine-1-carboxylate
N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indazole-3-carboxamide
ethyl({[4-(furan-2-yl)phenyl]methyl})(pyridin-2-ylmethyl)amine
4-{2-[2-(3-ethoxy-4-methoxyphenyl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
1-ethyl-4-(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)piperazin-2-one
N-[1-(1-methanesulfonylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
(3S,4S)-4-(propan-2-yloxy)-1-{2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carbonyl}pyrrolidin-3-ol
(3aS,6aS)-2-methyl-5-[(6-methylquinolin-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[(2-propyl-1,3-thiazol-4-yl)methyl]urea
N-[1-(4-fluorophenyl)ethyl]-2-methoxy-N-methylpyrimidine-5-carboxamide
1-(5-phenyl-1,2,4-oxadiazol-3-yl)azepan-4-amine
2-{4-[2-(8-methoxyquinolin-2-yl)-1H-imidazol-1-yl]-3,5-dimethyl-1H-pyrazol-1-yl}ethan-1-ol
N-cyclopropyl-4-methoxy-2-({1-[(2S)-pyrrolidine-2-carbonyl]piperidin-4-yl}oxy)benzamide
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(1H-1,2,4-triazol-3-yl)benzamide
3-cyclopropyl-5-[3-(2-fluorophenyl)-1H-pyrazol-5-yl]-1-methyl-1H-1,2,4-triazole
N-[phenyl(pyridin-4-yl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(2-methyl-1-benzofuran-7-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
propan-2-yl 3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
3-methyl-4-(2-{4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}ethoxy)-1,2,5-oxadiazole
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)[(2-phenoxypyridin-3-yl)methyl]amine
methyl 8-methyl-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-{2-oxo-2-[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethyl}imidazolidine-2,4-dione
2-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]-6-methylpyridin-3-ol
7-(4-chlorophenyl)-2-(5-cyclopropyl-1H-pyrazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(2-propyl-1,3-thiazole-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
7-[2-(oxan-2-ylmethoxy)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[5-benzoyl-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
4-{1-[(4-methylphenyl)methyl]-1H-1,3-benzodiazol-2-yl}-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(3-chloro-4-ethoxyphenyl)-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
3-{[1-(oxolane-2-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
4-[(2-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)methyl]morpholine
3-{1-[1-(thiophen-2-yl)ethyl]-1H-imidazol-2-yl}phenol
2-[1-(cyclohexylmethyl)-4-(1,2-oxazol-3-ylmethyl)piperazin-2-yl]ethan-1-ol
6-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}pyridine-3-carbonitrile