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5-methanesulfonyl-2-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine
2-amino-6-(3,4-dimethoxyphenyl)-4-[5-(hydroxymethyl)furan-2-yl]pyridine-3-carbonitrile
N-{2-[methyl(phenyl)amino]ethyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-{1-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-2-phenylethyl}-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
N-[2-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1H-imidazol-4-yl)ethyl]acetamide
(1,4-dioxan-2-ylmethyl)(methyl){[4-(trifluoromethoxy)phenyl]methyl}amine
N-[2-(pyridin-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
6-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-(1-ethylpiperidin-4-yl)-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]acetamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[(2R,3S)-2-amino-3-methylpentanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[(4-methylphenyl)methyl]-11-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[3-(cyclopentyloxy)propyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
N-[(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-3-yl)methyl]-1H-pyrrole-2-carboxamide
1-{5-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-ethyl-4-phenyl-9-(piperidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]butanamide
5-{2-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-(3-acetyl-1H-indol-1-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]butanamide
3-{2-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
N-[(4-chlorophenyl)(phenyl)methyl]-2-[methyl(piperidin-4-yl)amino]acetamide
N-(furan-2-ylmethyl)-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
(1S,2R)-N1-(2,1,3-benzothiadiazol-5-ylmethyl)-N2-tert-butyl-N1-methylcyclohexane-1,2-dicarboxamide
N-[(3S,4R)-1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[3-(4-fluorophenyl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(1-ethylpiperidin-4-yl)acetamide
3-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-7-fluoro-1,2-dihydroquinolin-2-one
{2-[(6-methoxypyridazin-3-yl)oxy]hex-5-en-1-yl}(methyl)(pyridin-3-ylmethyl)amine
4-{4-[2-(3-chlorophenyl)acetyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-[4-(methylsulfanyl)phenyl]urea
2-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
(1S,5R)-6-[(5-methylfuran-2-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
methyl 3-cyclobutaneamido-5-[(4-methylpentan-2-yl)amino]-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-(cyclopropylmethyl)-2-(4-oxo-4H-chromene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[5-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1,3-thiazol-2-yl]morpholine
3-chloro-N-cyclohexyl-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methylbenzamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-6-oxo-N-(oxolan-2-ylmethyl)-1,6-dihydropyrimidine-5-carboxamide
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
6-(4-benzyl-6-hydroxy-1,4-diazepane-1-carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 3-(cyclobutylmethoxy)-5-(2-methyl-1,4-oxazepane-4-carbonyl)benzoate
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-[4-(methylsulfanyl)benzoyl]piperidine
N,2-dimethyl-N-(2-methylprop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine
2-[5-(oxolan-2-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]pyridine
ethyl 4-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
1-[(3aS,6aS)-5-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-octahydropyrrolo[2,3-c]pyrrol-1-yl]propan-1-one
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]pentane-1,2-dione
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide