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2-methyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
{2-[(1R,5S,8S)-8-(dimethylamino)-3-azabicyclo[3.2.1]octane-3-carbonyl]pyridin-4-yl}methanol
N-ethyl-2-{4-[2-methyl-2-(morpholin-4-yl)propyl]piperazin-1-yl}pyrimidin-4-amine
2-{4-[4-(benzylsulfanyl)phenyl]-1H-pyrazol-1-yl}propanamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[3-(dimethylamino)benzoyl]-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
4-methyl-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]-1H-imidazole-5-carboxamide
2-{2-[(1-ethylpyrrolidin-3-yl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
3-{[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
N-[(6-{4-[1-(dimethylamino)ethyl]phenyl}pyridin-3-yl)methyl]acetamide
1-[(4-chlorophenyl)methyl]-N-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperidin-3-amine
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
3-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanamido)hexanoic acid
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(pyrrolidin-1-yl)butan-1-one
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(pyrimidin-4-ylmethyl)pyridin-2-amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(1-phenylethyl)propanamide
methyl[(4-methyl-1,3-thiazol-2-yl)methyl]{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
4-{1-oxaspiro[4.5]decan-3-yl}-4H-1,2,4-triazole
[5-({[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)furan-2-yl]methanol
3-[2-(2,3-difluorophenyl)acetyl]-N-(furan-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[3-(2-methylpropyl)-5-[2-(1H-pyrrol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]pyridine
3-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}propanoic acid
4-(4-acetylphenoxy)-1-cycloheptylpiperidine-4-carboxylic acid
4-[3-(1-ethyl-1H-pyrazol-3-yl)phenyl]pyridine
4-{3-[4-(dimethylamino)phenyl]propanoyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
2-(4-methyl-1H-pyrazol-1-yl)-1-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
7-{[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
2-methoxy-4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonitrile
6-methyl-2-{[3-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}quinolin-4-ol
4-ethyl-1-methyl-3-{1-[2-(1,2,3,6-tetrahydropyridin-4-yl)acetyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-N-cyclopropyl-2-acetamido-N-[(2-methoxyphenyl)methyl]pentanediamide
2-(3-hydroxypropyl)-9-(4-methylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{imidazo[1,2-a]pyridine-2-carbonyl}-1-[(4-methoxyphenyl)methyl]piperazin-2-one
3-(1-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidin-3-yl}-N-methylformamido)propanamide
N-cyclopropyl-5-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
2-{4-[(3-propoxypiperidin-1-yl)methyl]phenyl}-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
7-(1,3-benzothiazol-2-yl)-4-(2-methoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(4-fluorophenyl)-4-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}butanamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
6-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridin-3-amine
(4aS,8aR)-6-(pyrazin-2-yl)-1-(pyridin-2-ylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-{2-[1-(3-phenoxypropanoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylpyrazine-2-carboxamide
N-(oxolan-2-ylmethyl)-4-[2-(pyridin-4-yl)-1H-imidazol-1-yl]benzamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-5-methoxy-1-methyl-1H-indole-2-carboxamide
(3R,4S)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-3,4-dimethylpiperidin-4-ol
N-(adamantan-2-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide