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N-[(3-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]-3-(2-oxopyrrolidin-1-yl)propanamide
1-ethyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
1,1-dioxo-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1λ6-thiolane-3-carboxamide
2,2,6,6-tetramethyl-4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)piperidine
5,6-dimethyl-2-{2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
methyl({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[methyl(1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]ethan-1-ol
N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-{[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole
1-[3-(1H-imidazol-1-yl)propyl]-2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazole
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)urea
1-phenyl-4-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)-1H-1,2,3-triazole
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
N-ethyl-6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-3-carboxamide
(4aS,7aR)-1-[(6-ethoxyquinolin-2-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1r,4r)-4-methoxycyclohexyl]-3-(trifluoromethyl)benzamide
2-(3-methoxypropyl)-9-{thieno[3,2-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
2-(phenoxymethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
9-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylsulfamoyl)ethyl]-2,8-dimethylquinoline-4-carboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(1-propylcyclobutyl)methyl]-1,3-oxazole-4-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-methyl-6-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)pyrimidin-4-ol
1-benzyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
(3S,4R)-1-(6-aminopyridine-3-carbonyl)-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
N-[3-(3-chlorophenyl)phenyl]-1-[(3-hydroxyphenyl)methyl]piperidine-4-carboxamide
N-methyl-1-[(2-methylphenyl)methyl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-ethoxy-1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}ethan-1-one
3-(2-fluorophenyl)-3-phenyl-1-(thiomorpholin-4-yl)propan-1-one
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinolin-3-ylmethyl)benzamide
2-[(1S,5R)-3-[5-(methoxymethyl)furan-2-carbonyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-(adamantan-1-yl)-5-[(3S)-3-aminopiperidine-1-carbonyl]pyrimidin-4-ol
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-(piperidin-4-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
1-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
2-(2-fluorophenyl)-2-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}acetic acid
N-(2-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)benzamide
4-({4-methyl-5-[1-(pyridine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
4-{3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}-6-(propan-2-yl)pyrimidin-2-amine
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]thiophene-2-carboxamide
(3R,4R)-1-[(4-ethynylphenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
N-{[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
4-cyano-N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-1H-pyrrole-2-carboxamide
6-[4-(2-methoxyethoxy)piperidin-1-yl]-2-methylpyrimidin-4-amine
(2R,6S)-4-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-2,6-dimethylmorpholine
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]propanamide