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1-{1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-4-phenylpiperidin-4-yl}ethan-1-one
1-(but-2-yn-1-yl)-4-{1-[(3-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridine
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]morpholine-2-carboxamide
(1S)-2-cyclohexyl-1-[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-amine
6-methyl-2-[(4-methyl-1H-imidazol-5-yl)methyl]-5-[5-(1-methyl-1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
8-[(2S)-2-amino-3-(4-methoxyphenyl)propanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-oxo-4-phenylpiperazine-1-carboxamide
2-ethyl-N-[3-(pyridin-3-yloxy)propyl]pyrimidine-5-carboxamide
3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzonitrile
6-[(2,2-dimethyloxan-4-yl)amino]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
N-[2-oxo-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethyl]acetamide
(3S,9aR)-3-benzyl-2-methyl-8-(naphthalene-2-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(3-methoxy-2-propoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
(3R,9aR)-3-benzyl-8-(3,5-dichlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]quinoxaline
1-[(4-methoxyphenyl)methyl]-5-(3-methylfuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(methoxymethyl)-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,3-benzoxazole
2-(1H-1,3-benzodiazol-1-yl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methylpropanamide
N-[(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]acetamide
methyl 6-(3-cyclohexylpropanoyl)-2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-(3-{[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
3-(4-fluorophenyl)-3-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
3-({[(2-aminopyridin-3-yl)methyl]amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-{2-[4-(diphenylmethyl)piperazin-1-yl]-2-oxoethyl}-4-methylpiperazin-2-one
1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-(1,3,4-thiadiazol-2-yl)urea
6-chloro-2-(1-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
3-ethyl-1-(4-fluoro-3-methylphenyl)-3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]urea
N-[(4-fluorophenyl)methyl]-N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-cyclopentyl-6-[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
8-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(2R,6R)-4-{3-[(2-methoxyethyl)(methyl)amino]propanoyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
ethyl 2-(1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-2-yl)acetate
6-(diethylamino)-1-(2-propoxyethyl)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
1-{4-[5-(2-ethylpiperidine-1-carbonyl)-2-methoxyphenoxy]piperidin-1-yl}ethan-1-one
3-(2-phenylpropyl)-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-tert-butyl-4-[4-(3-chloropyridin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
3-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
5-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-1-methyl-1,2-dihydropyridin-2-one
5-(ethoxymethyl)-1-(2-phenylethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
(3S,4R)-N,N-dimethyl-1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]-4-(propan-2-yl)pyrrolidin-3-amine
N-benzyl-1-methyl-5-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-(morpholine-4-carbonyl)piperidine-4-carboxylic acid
6-methoxy-3-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
4-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-chlorophenol