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9-[(5-ethylpyridin-2-yl)methyl]-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[1-(4-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyrimidin-2-one
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
2-[4-(furan-2-ylmethyl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
8-(5-ethyl-1,3-oxazole-4-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]oxy}benzamide
methyl[2-(oxan-2-yl)ethyl]{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanoic acid
(2R,3S,6R)-5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-methyl-N-(pyridin-3-ylmethyl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
N'-cyclopentyl-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]butanediamide
3-methyl-7-[2-(4-phenylphenyl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-hydroxypropanamide
3-{[1-(1,1-dioxo-1λ6-thiane-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
(3aR,6aR)-2-methanesulfonyl-5-{[5-(methylcarbamoyl)furan-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(4-methylphenyl)methyl]piperazin-2-one
(2S,4R)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
3-(cyclopentylsulfamoyl)-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N4,N4,5-trimethyl-N2-[4-(morpholin-4-yl)butan-2-yl]pyrimidine-2,4-diamine
1-[2-(dimethylamino)-4-{[(2-methyloxolan-2-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
8-[3-(pyridin-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(pyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(3R,4R)-1-(3-ethoxybenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
(4aS,7aR)-1-(3-ethoxybenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-imidazole
8-[(3-hydroxyphenyl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-2-(phenoxymethyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2-(pyrrolidin-3-yl)benzamide
N-[(2-chlorophenyl)methyl]-3-[2-(trifluoromethyl)morpholin-4-yl]propanamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
propan-2-yl 2-chloro-5-[(3-methoxypiperidine-1-carbonyl)amino]benzoate
3-methyl-5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
4-fluoro-N-[(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]benzamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
N-[1-(3,4-dimethylphenyl)ethyl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(2-methoxyethyl)-4-{[2-(pyrrolidin-1-yl)ethyl]sulfamoyl}benzamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]ethan-1-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}propanamide
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
1-(cyclopropylmethyl)-3-({[(3,5-difluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
4-chloro-N,N-dimethyl-5-{[4-(3-methylpyridin-4-yl)piperazin-1-yl]methyl}-1,3-thiazol-2-amine
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
2-{[4-(2,3,4-trimethoxyphenyl)phenyl]sulfanyl}acetamide
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
6-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-methylpyrimidin-4-amine
(2-{[(4-methanesulfonylphenyl)methyl][(2-methylphenyl)methyl]amino}ethyl)dimethylamine
9-(2,3-dihydro-1H-inden-1-yloxy)-4-(1,3-thiazole-5-carbonyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 4-(2-methoxyethyl)-1-(3-methylthiophene-2-carbonyl)piperidine-4-carboxylate