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2-(2,2-diphenylethyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]morpholine
{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amine
7-(1-benzothiophen-3-yl)-4-(1,2-oxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1R,9aR)-1-[4-(pyridin-4-yl)piperazine-1-carbonyl]-octahydro-1H-quinolizine
2-(2,4-dichlorophenoxy)-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]acetamide
4-methyl-N-[(1R,3S)-3-[(oxan-4-yl)carbamoyl]cyclopentyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
(3S,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]morpholine-4-sulfonamide
N-[3-(4-fluorophenyl)phenyl]-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
N-[2-(pyridine-3-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
N,N-dimethyl-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-(1-hydroxy-2-methylpropan-2-yl)-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
methyl 1-(2-methoxyethoxy)-2-oxo-8-(5-phenoxyfuran-2-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-3-(1H-1,3-benzodiazol-2-yl)propan-1-one
7-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2,3-dimethyl-1H-indole
1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
N-(2,4-dimethoxyphenyl)-3-{1-[(2R)-pyrrolidine-2-carbonyl]piperidin-4-yl}propanamide
3-[4-(2-cyclopropylacetyl)-6-hydroxy-1,4-diazepan-1-yl]pyrazine-2-carbonitrile
6-methyl-2-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)quinolin-4-ol
1-(4-cyclopentyl-6-hydroxy-1,4-diazepan-1-yl)-2-(thiophen-2-yl)ethan-1-one
3-[(3S,4R)-4-(dimethylamino)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-N-[2-(1H-indol-3-yl)ethyl]propanamide
N-[4-(dimethylamino)phenyl]-3-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propanamide
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,5,6-trimethylpyridine-3-carboxamide
2-{1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1,4-diazepan-6-yl}acetic acid
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(prop-2-en-1-yl)amino]-N-[(2-fluorophenyl)methyl]acetamide
(1R,5R)-6-(cyclopropylmethyl)-3-[4-(piperidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}({[5-(methoxymethyl)furan-2-yl]methyl})methylamine
4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-6-methyl-1,2-dihydropyridin-2-one
1-ethyl-4-{[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]methyl}-3,5-dimethyl-1H-pyrazole
dimethyl[({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methyl)sulfamoyl]amine
2-{1-cyclohexyl-5-[3-(4-methylpiperazin-1-yl)butyl]-1H-1,2,4-triazol-3-yl}acetamide
2-(4-chloro-1H-pyrazol-1-yl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}propanamide
N,2-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
8-[2-(dimethylamino)acetyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-fluoro-7-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(3,3,3-trifluoropropanoyl)piperidine-2-carboxamide
methyl N-(2-oxo-2-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethyl)carbamate
1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(furan-2-yl)-1H-pyrazol-5-yl]piperidine
N-[1-ethyl-2-(2-fluorophenyl)-7-(5-oxo-1,4-diazepane-1-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
ethyl 1-[(3-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
2-chloro-6-methoxy-4-[1-(oxolan-2-ylmethyl)-1H-imidazol-2-yl]phenol
3-(3-methoxyphenyl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1H-pyrazole-4-carboxamide
(2R,3R,6R)-5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{[1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1H-1,2,3,4-tetrazole
5-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-5-oxopentanamide
N-(3,4-dimethylphenyl)-3-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}propanamide
N,1-dimethyl-N-(1,2-oxazol-3-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[(1R,2R)-2-hydroxycyclohexyl]methyl}-5-methyl-3,4-dihydroquinazolin-4-one