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N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-(4-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[3-(1H-1,2,3-triazol-1-yl)propyl]acetamide
1-(3,5-dimethylphenyl)-4-[5-(methoxymethyl)thiophene-2-carbonyl]piperazin-2-one
1'-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2,4-dimethyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]pyrimidine-5-carboxamide
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(6-methylpyridazin-3-yl)-decahydro-1,6-naphthyridin-2-one
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N-{3-[methyl(phenyl)amino]propyl}-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
N-(furan-2-ylmethyl)-2-[(3-methoxyphenyl)amino]butanamide
1-(1-phenyl-1H-pyrazol-5-yl)-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
3-[(dimethylamino)methyl]-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidin-3-ol
2-ethyl-N,6-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-4-amine
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-(3-fluoro-5-methylphenyl)urea
4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(2-methoxyethoxy)-1-[4-(4-methylphenoxy)piperidin-1-yl]ethan-1-one
(3S,4S)-1-(2,5-dimethylfuran-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
3-{[(1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
(4aS,8aS)-2-({2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}methyl)-decahydro-2,7-naphthyridin-4a-ol
ethyl 4-[(2S,4S)-4-amino-2-(methylcarbamoyl)pyrrolidin-1-yl]piperidine-1-carboxylate
6-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[4-(methylsulfanyl)phenyl]methyl}-N-(prop-2-en-1-yl)but-3-enamide
N-ethyl-2-(6-methoxypyridin-3-yl)pyrimidin-4-amine
N-[2-(dimethylamino)ethyl]-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propanamide
1-(3-cyanopyridin-2-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
4-ethyl-3-(piperidin-3-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[4-(2-ethylphenyl)piperazin-1-yl]-N-(2-methylphenyl)-3-oxopropanamide
3-{[(4-fluorophenyl)methyl]amino}-N-[3-(propan-2-yloxy)propyl]benzamide
2-[1-(2,2-dimethylpropyl)-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl]ethan-1-ol
3-methyl-8-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S)-2-amino-3-hydroxy-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
3-{3-[(4-hydroxyphenyl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl}propanoic acid
(2S,4S)-N-methyl-4-(4-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
N-butyl-N,5-dimethyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-phenylpiperazine
{1-[5-(aminomethyl)pyridin-2-yl]-3-propylpiperidin-3-yl}methanol
1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide
3-cyclopentyl-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-(thiophen-3-ylmethyl)urea
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
4-(1-methyl-1H-imidazol-2-yl)-1-(5-methyl-4-phenylthiophene-3-carbonyl)piperidine
5-chloro-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-3-carboxamide
4-ethyl-1-methyl-3-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]propyl}-3,4-dihydroquinazolin-4-one
6-(2H-1,3-benzodioxol-5-yl)pyridin-2-ol
2-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
7-chloro-2-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-3-methyl-1H-indole
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]-1H-pyrazole-4-carboxamide