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2-methyl-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,4-diazepan-5-one
N-(4-chloro-2-fluorophenyl)-2-(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)acetamide
1-({5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]furan-2-yl}methyl)-4-methylpiperazine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(4S)-3,3,4-trimethyl-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-ol
N,N-dimethyl-8-oxo-7-(prop-2-en-1-yl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-cyclopropyl-3,5-dimethoxy-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
methyl 5-[(furan-3-ylmethyl)amino]-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
9-(2,4-dimethylpyrimidine-5-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]propan-1-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-4-ol
3-{[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]methyl}-5-(oxolan-2-yl)-1,2,4-oxadiazole
N-(2-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}ethyl)methanesulfonamide
4-(2-methylquinolin-4-yl)-2-[(4-phenylpiperazin-1-yl)methyl]phenol
2-(3-methylphenyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyrimidin-4-ol
N-[2-(morpholin-4-yl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
3-{[1-(adamantan-2-yl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-methyl-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(1,2,3,4-tetrahydronaphthalen-1-yl)urea
2-amino-N-{2-fluoro-4-[3-(trifluoromethyl)phenyl]phenyl}acetamide
2-[4-(hydroxymethyl)-4-[(4-methoxyphenyl)methyl]piperidin-1-yl]pyridine-3-carboxamide
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-1H-indole-3-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
4-[(diethylamino)methyl]-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-ethylfuran-2-carboxamide
2-(2-hydroxyethyl)-9-(trimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-{[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]formamido}ethyl)pyridine-3-carboxamide
1-(5-cyclopropyl-1H-pyrazole-3-carbonyl)-4-(1H-imidazol-2-yl)piperidine
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
(1R,2R)-2-{ethyl[(8-methoxyquinolin-2-yl)methyl]amino}cyclohexan-1-ol
N-[1-(1H-pyrazol-1-yl)propan-2-yl]quinoxaline-5-carboxamide
1-cyclopentanecarbonyl-N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-amine
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]pyrrolidin-3-yl]urea
3-{2-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-cyclopropyl-5-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-phenyl-1H-1,2,4-triazole
N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
4-methyl-2-[1-(1H-1,2,3-triazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-(2,3-dihydro-1-benzofuran-7-carbonyl)-4-(hydroxymethyl)piperidin-4-ol
5-{[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]methyl}-2-methoxybenzoic acid
9-(2-ethylpyrimidine-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(pyridin-3-yl)-5-[4-(2,2,2-trifluoroethyl)piperazine-1-carbonyl]pyrimidin-4-ol
3-benzyl-8-(1-methoxypropan-2-yl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[3-(pyridin-2-yl)azetidine-1-carbonyl]-2-(trifluoromethyl)-1H-1,3-benzodiazole
N-(2-methylpropyl)-1-[(1s,4s)-4-(2-methyl-1,3-thiazole-4-amido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-(6-phenylpyridine-2-carbonyl)-1,4-oxazepan-6-ol
2-(2-{4-[(2-fluoro-3-methoxyphenyl)methyl]piperazin-1-yl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one