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N-{1-[1-(2,2-dimethylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
2-{[2-(oxan-2-yl)ethyl]amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-1,2-dihydroisoquinolin-1-one
5-hydroxy-N-propyl-N-(pyridin-4-ylmethyl)pyrazine-2-carboxamide
2,4-dimethyl-N-[4-(4-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}piperidin-1-yl)phenyl]benzamide
2-[1-methyl-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol
N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
6-ethyl-3-[1-(pyrazin-2-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-(2-hydroxybenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 6-(3-hydroxyphenyl)pyridine-3-carboxylate
N-(1-benzylpyrrolidin-3-yl)-3-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]propanamide
N-[3-(pyridin-3-yloxy)propyl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-5-(thiophen-2-yl)-1,2,4-oxadiazole
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-3-yl]acetamide
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-3-phenoxypropan-1-one
6-(2-chlorophenyl)-N-(2-hydroxy-3-methoxypropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}cyclohexane-1-carboxamide
4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine-1-sulfonamide
1-[4-(3-hydroxy-3-methylbutyl)benzamido]cycloheptane-1-carboxamide
3-[3-(benzyloxy)azetidine-1-carbonyl]-1-ethyl-3-methylpiperidine
1-[3-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]pyrrolidin-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-5-ylmethyl)acetamide
1-[4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenyl]imidazolidin-2-one
N,N-dimethyl-5-{[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]methyl}pyridin-2-amine
3-[({1-[(3-chloro-2,4-difluorophenyl)methyl]piperidin-4-yl}oxy)methyl]pyridine
6-methyl-4-[3-(trifluoromethyl)phenyl]-2,3-dihydropyridazin-3-one
4-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-2-phenylpiperazine
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[(5-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
ethyl 5-[(3-methoxyphenyl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
8-(1-ethylpiperidin-4-yl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(1H-indol-1-ylmethyl)-N-[1-(1,3-thiazol-2-yl)propyl]-1H-pyrazole-3-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-(4-methylphenyl)quinoline-4-carboxamide
2-butyl-8-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}thiophene-2-carboxylic acid
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(4aS,8aR)-6-[3-(methylsulfanyl)propyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
7-(5-methylthiophen-2-yl)-4-(1H-pyrrole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclopropyl-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-4-carboxamide
2-{4-[2-(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)ethyl]-1,3-thiazol-2-yl}pyrimidine
(2,1,3-benzoxadiazol-4-ylmethyl)(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
(4aS,8aR)-1-(3-aminopropyl)-6-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
5-(furan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 5-{[(3,4-difluorophenyl)methyl]amino}-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,4R)-1-(cyclopentylcarbamoyl)-4-phenylpyrrolidine-3-carboxylic acid
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(pyridin-3-yloxy)ethan-1-one