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N4-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-methylpyrimidine-2,4-diamine
3-{1-[2-(diethylamino)ethyl]-1H-imidazol-2-yl}phenol
N-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
4-methyl-2-{2-[3-(1-methylpiperidin-3-yl)propanamido]ethyl}-1,3-thiazole-5-carboxylic acid
9-[(2R)-2-amino-3-phenylpropanoyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(quinolin-8-yloxy)methyl]-N-(1H-1,2,4-triazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
1-{1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
N-cyclopentyl-5-(1H-indazole-3-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-methyl-N-[(1-methylpiperidin-3-yl)methyl]-2-oxo-2,3-dihydro-1,3-benzoxazole-6-sulfonamide
[(1-ethyl-1H-imidazol-2-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
4-chloro-1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-3-carboxamide
(3S,4R)-4-(hydroxymethyl)-1-{[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-3-ol
3-{[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)amino}propane-1,2-diol
(1S,4S)-2-(3-chlorophenyl)-5-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-2-(thiophen-3-yl)acetamide
4-{1-[1-(4,5-dimethylthiophene-2-carbonyl)piperidin-4-yl]ethyl}morpholine
2-(2-{[4-(dimethylcarbamoyl)piperazin-1-yl]methyl}phenoxy)propanoic acid
1-[1-(4-methylbenzoyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
2-hydroxy-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-4-(methylsulfanyl)butanamide
5-{2-[(prop-2-en-1-yl)amino]ethyl}-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(3-methylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{4-[(1H-imidazol-2-ylmethyl)(methyl)carbamoyl]phenyl}-5-methylfuran-2-carboxamide
3-[5-(2,3-dihydro-1-benzofuran-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-({5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-benzyl-1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
6-[ethyl(methyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-phenyl-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
3-(dimethylamino)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}benzamide
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-(pyrrolidine-1-carbonyl)pyrrolidine-2-carboxylic acid
1-{4-[3-({[(2,3,6-trifluorophenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
6-chloro-N,N-dimethyl-3-[({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[2-(dimethylamino)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-6-(morpholine-4-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}spiro[2.2]pentane-1-carboxamide
({6,7-dimethoxy-2-[(4-methylphenyl)methoxy]quinolin-3-yl}methyl)(1,4-dioxan-2-ylmethyl)amine
4-ethyl-5-methyl-N-[2-(pyridin-3-yl)ethyl]thiophene-3-carboxamide
5-{[2-(furan-2-yl)phenyl]methyl}-4-(furan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
7-(7-chloro-4-hydroxyquinoline-3-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl})amine
1-(4-fluoro-3-methoxyphenyl)-3-(2-hydroxyethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
ethyl 4-[(4-chlorophenyl)methyl]-1-[3-(pyrazin-2-yl)propanoyl]piperidine-4-carboxylate
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(2-fluorobenzoyl)piperidin-3-yl]piperazine
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
N,2-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(4-methanesulfonylphenyl)ethyl]-3-(1H-pyrazol-4-yl)benzamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-ethylpyrimidine-5-carboxamide
{2-fluoro-5-[6-(piperazin-1-yl)pyridin-2-yl]phenyl}methanol
N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-4-methanesulfonylpiperazine-1-carboxamide