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N-[3-(3,4-dimethoxyphenyl)propyl]-3-phenyl-1H-pyrazole-4-carboxamide
N,N-bis(pyridin-3-ylmethyl)-3-(pyridin-4-yl)propanamide
1-(5-phenyl-1,2-oxazole-3-carbonyl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
2-(cyclopropylmethyl)-9-[(3,4-dimethoxypyridin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(2-fluorophenyl)ethyl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-ethyl-1-(naphthalene-2-carbonyl)-1,4-diazepan-5-one
5-ethyl-2,3-dimethyl-N-(quinolin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-amino-3-ethyl-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
5-fluoro-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyrimidin-4-amine
2-(2-chlorophenyl)-3-methyl-N-(1,2-oxazol-5-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
(2H-1,3-benzodioxol-4-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-(quinazolin-4-yloxy)ethan-1-one
2-(dimethylamino)-N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-2-(2-methylphenyl)acetamide
2-fluoro-5-sulfamoyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2,2-dimethylpropan-1-one
methyl 6-(1-phenylcyclopropanecarbonyl)-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(2H-1,3-benzodioxol-5-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}ethan-1-one
4-[1-(2-methoxyphenyl)-5-(oxan-4-yl)-1H-1,2,4-triazol-3-yl]pyridine
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl][(4-methoxyphenyl)methyl]methylamine
1,3-dimethyl-N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)-1H-pyrazole-5-carboxamide
N-methyl-3-[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanamide
3-(1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)pyridine
(1S,6R)-3-methyl-9-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
(1R,7S)-N-methyl-4-oxo-3-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
[(2S,6S)-4-(1H-pyrrole-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
1-cyclopentyl-4-[2-(phenylamino)pyrimidine-5-carbonyl]piperazin-2-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(4-{[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenyl)acetamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(4-fluorophenoxy)piperidine
7-(cyclohexylmethyl)-2-[3-(pyridin-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
6-fluoro-4-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
1-[3-(3-fluorophenyl)phenyl]-N-(oxan-3-yl)piperidin-4-amine
N-[2-(dimethylamino)ethyl]-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N2-(4-methylphenyl)-6-[4-(piperidine-1-carbonyl)phenyl]-1,3,5-triazine-2,4-diamine
3-cyclopropyl-5-[1-(4-methyl-1H-pyrazol-1-yl)ethyl]-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-2-amine
3-methyl-5-{2-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-({[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)amino)propan-2-ol
3-({1-[(2-chloro-6-fluorophenyl)methyl]-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl}methyl)imidazolidine-2,4-dione
N-(2,2-diphenylethyl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
methyl 5-(4-methylpyrimidin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(2-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-{1-[7-(cyclohexylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}-2-methoxyacetamide
5-(5-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}furan-2-yl)-1H-pyrazole
2-cyclopropyl-N-(pyrimidin-4-ylmethyl)-1,3-benzoxazole-6-carboxamide