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1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}azetidin-3-ol
(3S,4R)-4-(3-methoxyphenyl)-1-(quinolin-6-ylmethyl)pyrrolidine-3-carboxylic acid
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(3,4-difluorophenyl)methyl]acetamide
methyl (1R,3S,3aR,6aS)-3-(4-butoxyphenyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
4-methoxy-6-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-2-amine
N-benzyl-3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
4-{4-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
7-[(3-methoxyphenyl)methyl]-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
1-(4-fluorophenyl)-4-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)piperazine
(1R,5S,6S)-6-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-azabicyclo[3.1.0]hexane
3-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
N-butyl-N-[(2-fluorophenyl)methyl]-3-methanesulfonamidopropanamide
2-(2-chloro-4-fluorophenyl)-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
N-(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}phenyl)ethane-1-sulfonamide
2-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(furan-2-yl)pyrimidine
4-{2-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,2,4-trimethylpyrimidine-5-carboxamide
6-(2-chlorophenyl)-N-(1-hydroxybutan-2-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-{2-[1-(2-methylfuran-3-carbonyl)piperidin-2-yl]ethyl}morpholine
(1R,5R)-N,N-dimethyl-6-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(1S,5R)-3-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]propan-1-one
N-(2,4-dimethylphenyl)-3-{octahydropyrrolo[1,2-a]piperazin-2-yl}-3-oxopropanamide
ethyl(methyl)[2-methyl-3-(5-methyl-4-phenyl-1H-imidazol-1-yl)propyl]amine
N'-[(4-methoxyphenyl)methyl]-N'-(2-methylpropyl)pentanediamide
1-{4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}-3-(pyridin-4-yl)propan-1-one
N-butyl-N-[(3-methoxyphenyl)methyl]piperidine-3-carboxamide
(1R,3s,6r,8S)-4-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-4-azatricyclo[4.3.1.13,8]undecane
7-fluoro-N,3-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-benzofuran-2-carboxamide
7-(2-cyclohexylethyl)-2-(5-methyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-(4-cyclohexylpiperazine-1-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
8-(6-methoxypyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]methyl}-4-(4-fluorophenyl)piperazine
N-methyl-5-{[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamido]methyl}furan-2-carboxamide
1-[(2S,4R)-1-[(4-methoxynaphthalen-1-yl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
2-[2-(dimethylamino)ethyl]-9-(4,6-dimethylpyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-ethoxy-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}pyrimidin-2-amine
4-({[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl](methyl)amino}methyl)-1-cyclopentylpyrrolidin-2-one
5-{4-[3-(methylsulfanyl)-1H-1,2,4-triazol-5-yl]phenyl}imidazolidine-2,4-dione
2-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-4-carboxamide
N,N,4-trimethyl-5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrimidin-2-amine
2-methyl-5-({3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-1,3-benzothiazole
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
6-fluoro-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide