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(4aS,8aR)-6-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(oxolan-2-ylmethyl)-9-(1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
5-methyl-3-[5-(thiophene-2-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
5-{2-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
methyl 4-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
4-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
(1R,9S)-5-amino-12-methyl-3-[4-(prop-2-en-1-yloxy)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
3-[1-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-1-ol
2-(2-hydroxyethyl)-8-[2-(3-methoxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(difluoromethyl)-5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrazole
N-cyclopentyl-2,4-dimethoxy-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzamide
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
2-(1-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}piperidin-2-yl)pyridine
3-(piperidine-1-carbonyl)-2-(3,4,5-trimethoxyphenyl)pyridine
4-({N-ethyl-1-[2-(ethylamino)pyrimidin-5-yl]formamido}methyl)benzoic acid
1-(2-oxo-2-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-(5-chloropyridin-2-yl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-(4-chloro-2-fluorobenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-amino-3-(3,4-dimethoxyphenyl)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
(1S,5R)-6-(1H-imidazol-2-ylmethyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
(3aS,6aS)-2-(3-cyano-5,6,7,8-tetrahydroquinolin-2-yl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-fluoro-N-(3-hydroxypropyl)-N-[(2-methoxyphenyl)methyl]-3-methyl-1H-indole-2-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-1,2-oxazole-3-carboxamide
(2S,4R)-4-amino-1-[(5-ethylpyridin-2-yl)methyl]-N-methylpyrrolidine-2-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxybenzamide
{2-[3-chloro-5-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}methanol
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
4,6-dimethyl-2-oxo-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-methoxy-6-(2,4,6-trimethylphenyl)pyrimidin-2-amine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]pyrimidin-2-amine
3-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydropteridin-4-one
1-cyclohexyl-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
7-(propan-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(3R,4R)-1-(5-chloro-3-fluoropyridin-2-yl)-4-ethylpiperidine-3,4-diol
methyl 3-(pyrazine-2-amido)-5-[(quinolin-2-ylformamido)methyl]benzoate
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propan-1-one
1-(4,6-dimethylpyrimidin-2-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]piperidin-4-amine
1-ethyl-N-[2-(2-fluorophenyl)ethyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-({[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylpropanamide
N-ethyl-1-(2-methylpropyl)-4-oxo-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-(piperidine-1-carbonyl)pyrazine
5-{[methyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})amino]methyl}pyrimidin-2-amine
2-amino-4-[2-(dimethylamino)pyrimidin-5-yl]-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(4-methoxyphenyl)-4-[3-(2-methyl-1H-indol-1-yl)propanoyl]piperazin-2-one
1-ethyl-3,5-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazole-4-carboxamide