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2-(2H-1,3-benzodioxol-5-yloxy)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)thiophene-3-carboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
5-methanesulfonyl-2-methyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]pyrimidin-4-amine
2-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(pyrazin-2-ylmethyl)amine
6-(3-oxo-3-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propyl)-2,3-dihydropyridazin-3-one
5-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-2-(methoxymethyl)pyrimidine
2-(3-methoxyphenyl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)azetidine
3-[(4aR,7aS)-6,6-dioxo-4-(4,4,4-trifluorobutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-5-[5-(2-methylpropyl)-1,2-oxazol-3-yl]-1H-1,2,4-triazole
[1-(1H-imidazol-1-yl)propan-2-yl]({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl})amine
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
2-propyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,3-thiazole-4-carboxamide
N-cyclohexyl-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
N,1-dimethyl-2,4-dioxo-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-indazole-3-carboxamide
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(3-phenoxyphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-3-(3-methoxypyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
[(3R,4R)-1-[4-(1H-imidazol-1-yl)benzoyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-cyclopropyl-5-[1-(dimethyl-1H-1,2,4-triazol-1-yl)propan-2-yl]-1-(4-methoxyphenyl)-1H-1,2,4-triazole
8-(4-hydroxybutyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(1R,5R)-3-(2-chlorobenzoyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,5R)-6-[2-(phenylsulfanyl)ethyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(2,4,5-trimethoxyphenyl)methyl]-3,9-diazaspiro[5.6]dodecan-10-one
3-[({1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-yl}oxy)methyl]pyridine
2-(2-chloro-6-fluorophenyl)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
1-[4-phenyl-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethan-1-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(2,5-dioxoimidazolidin-4-yl)acetamide
N-[(2,5-difluorophenyl)methyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
ethyl({[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(3-phenylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[(3R,4R)-1-[(4-ethylphenyl)methyl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
(1R,2R)-N-[2-(4-methylpiperazin-1-yl)ethyl]-2-phenylcyclopropane-1-carboxamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[(5-methylpyrazin-2-yl)methyl]propanamide
N-benzyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-(2-phenylethyl)acetamide
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(2-methylphenyl)piperidine
4-(2-methoxypyridin-3-yl)-6-(4-methyl-1H-pyrazol-1-yl)pyrimidine
4-[1-(4-carboxybutyl)piperidin-3-yl]benzoic acid
4-[(3-chlorophenyl)methyl]-1-[(2-ethoxyphenyl)methyl]-1,4-diazepan-5-one
1-(2-methoxyphenyl)-2,2-dimethyl-4-(2-methyloxane-2-carbonyl)piperazine
1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
(3aR,6aS)-5-(1-benzyl-1H-pyrazole-4-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(2-hydroxybenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]pyrimidin-5-yl}acetic acid
[(3R,4S)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}pyrazine