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[(2-chloro-6-fluorophenyl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
1-ethyl-4-[({5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)methyl]pyrrolidin-2-one
2-(1H-pyrazol-1-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]butan-1-one
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-benzyl-3-butyl-1-{2-[(3R)-3-methylpiperazin-1-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-cyclopropyl-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N,N-dimethyl-2-({[4-(trifluoromethyl)pyrimidin-2-yl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N-(2,5-dimethylphenyl)-3-{[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}propanamide
4-({2-[(3-methylpyridin-2-yl)amino]ethyl}amino)-N-(propan-2-yl)pyridine-2-carboxamide
N-cyclopropyl-2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]pyridine-4-carboxamide
(2S)-2-amino-1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-(1H-imidazol-4-yl)propan-1-one
(3S,4R)-3-benzyl-1-(6-methoxypyrimidin-4-yl)-4-methylpiperidin-4-ol
1-(3-chlorophenyl)-4-[1-(1-ethylpiperidine-4-carbonyl)piperidin-3-yl]piperazine
2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)benzene-1,3-diol
N-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-3-methylbut-2-en-1-one
6,6-dimethyl-N-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(2-methoxyethyl)-N'-(3-methylphenyl)-N-(thiophen-2-ylmethyl)propanediamide
1-[2-(4-methoxy-3-methylphenyl)pyrimidin-4-yl]pyrrolidin-3-ol
ethyl 4-[(3-methoxyphenyl)methyl]-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carboxamide
8-(1,3-thiazol-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-3-ol
(1S,3R)-3-amino-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}cyclopentane-1-carboxamide
N-[3-(furan-2-yl)propyl]-2-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-oxoacetamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(2-{2-[1-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
(2S,4S)-N-ethyl-1-(furan-3-ylmethyl)-4-[3-(pyridin-4-yl)propanamido]pyrrolidine-2-carboxamide
N-[4-(2-methyl-6-propylpyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-5-ethyl-2-methylpyrimidin-4-amine
N-methyl-N-(2-phenylethyl)-1-(pyridine-3-sulfonyl)piperidin-3-amine
2-(2-methyl-1,3-thiazol-4-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
3-cyclopropyl-1-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
5-(2,6-dimethoxyphenyl)-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,2,4-triazin-3-amine
[(3R,4R)-4-[(dimethylamino)methyl]-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-3-yl]methanol
6-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
N-[3-(1H-indol-2-yl)phenyl]-1-[2-(methylsulfanyl)acetyl]piperidine-3-carboxamide
6-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
4-{5-[(4-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
N-(1-{2-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(2-methoxyphenyl)acetamide
3-methoxy-6-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridazine
N-cycloheptyl-2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoacetamide
2-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3-methyl-1-phenyl-1,2-diazinane
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(1,3-thiazol-2-yl)piperidine
N-methyl-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
N-butyl-N-(furan-2-ylmethyl)-1H-1,3-benzodiazole-2-carboxamide
6-methyl-2-({2-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}sulfanyl)-3,4-dihydropyrimidin-4-one