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N-(1-carbamoylcyclopentyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
5-(1-cyclopropanecarbonylpyrrolidin-2-yl)-N-(2,3-dihydro-1H-inden-4-yl)thiophene-2-carboxamide
1-(3-{3-[3-(1-methyl-1H-pyrazol-4-yl)phenyl]-1H-pyrazol-1-yl}propyl)piperidine
2-amino-N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-methyl-1,3-benzothiazole-6-carboxamide
2-[1-(2-fluorophenyl)-5-(2-methoxypyridin-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-(1-{1-[(2S)-2-aminobutanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-methoxybenzamide
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-5-[(methylsulfanyl)methyl]furan-2-carboxamide
N-{[1-(cyclopentylmethyl)piperidin-3-yl]methyl}-4,4,4-trifluorobutanamide
N-(2,3-dihydroxypropyl)-5-(2,5-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-4-(3-hydroxy-3-methylbutyl)benzamide
2-ethyl-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
N-methyl-4-[3-(3-methylpyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
8-(4-ethoxybenzenesulfonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl 3-{[1-(cyclopropylmethyl)-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
(5-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-indol-2-yl)methanol
N-cyclohexyl-3-{[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}propanamide
N-[2-(2-chlorophenoxy)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]pyridine-3-carbonitrile
2-{[2-(trifluoromethyl)phenyl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
(1,4-dioxan-2-ylmethyl)(methyl){[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-methyl-2-(2-oxoimidazolidin-1-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]acetamide
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-4-yl)propan-1-one
ethyl 4-{6-benzoyl-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
5-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
5-(1-tert-butyl-1H-pyrrol-3-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-[1-(3-chlorobenzenesulfonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
9-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
methyl 2-[3-(4-chlorophenyl)-3-phenylpropanamido]acetate
[(2-chloro-6-fluoro-3-methoxyphenyl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-[2-(2-methylphenyl)ethyl]piperidine
N-[1-(pyrazin-2-yl)piperidin-4-yl]-2-(pyrrolidin-3-yl)benzamide
6-chloro-N-(3-hydroxypropyl)-2-methyl-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
2-acetyl-8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(1,4-dioxan-2-ylmethyl)-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-4-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]butan-1-one
1-[2-(cyclohex-1-en-1-yl)ethyl]-2-(propan-2-yl)-1H-imidazole
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
1-[3-(benzyloxy)piperidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[2-(pyridin-4-yl)ethyl]amine
[2-(2,4-dimethylphenoxy)ethyl](methyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
(1S,5R)-N,N-dimethyl-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-sulfonamide
7-(2-phenoxyacetyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2R,3R)-3-amino-1'-(4-hydroxy-3-methylbenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(1R,2R,6S,7S)-4-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)-4-azatricyclo[5.2.1.02,6]decane
N1,N1-dimethyl-N3-{[5-(methylcarbamoyl)furan-2-yl]methyl}piperidine-1,3-dicarboxamide
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
2-methyl-N-(oxan-3-yl)-7-(1H-pyrrole-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine