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(3S,9aR)-8-{[3-(methylsulfanyl)phenyl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(2-fluorophenoxy)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(methylsulfanyl)acetamide
(2S,4S)-4-amino-1-[5-(methoxymethyl)thiophene-2-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(3-methylbut-2-en-1-yl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-cyclopropyl-5-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
7-(cyclopropylmethyl)-2-(4-methyl-1H-imidazole-2-carbonyl)-2,7-diazaspiro[4.5]decane
2-[5-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]acetic acid
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazine
2-(2-ethyl-1H-imidazol-1-yl)-1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
(2R,4S)-1-[(2,4-dimethoxyphenyl)methyl]-4-hydroxypiperidine-2-carboxylic acid
N-(3-cyano-4-methoxyphenyl)-4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carboxamide
4-[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-imidazol-2-one
N,N-dimethyl-4-{[2-(propylamino)pyrimidin-5-yl]methyl}piperazine-1-carboxamide
4-[7-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
13-[3-(1H-pyrazol-1-yl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]propanamide
3-{[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]methyl}benzoic acid
N-cyclopropyl-4-methoxy-3-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[(4-fluorophenyl)methyl]-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-ethyl-N,3-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]piperidine-3-carboxamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(pyrrolidine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[2-(1H-indol-1-yl)ethyl]-N,2-dimethyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-({[1-(3-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyrimidine
1-(1H-imidazol-2-ylmethyl)-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-1,2,3-triazole
3-{1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}piperidine
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[(2R)-pyrrolidine-2-carbonyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2,6-dimethyl-5-(2-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
4-methyl-5-(prop-2-en-1-yl)-6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidin-2-amine
(1R,5S)-6-methyl-3-(4-methyl-1H-imidazole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-cyclohexyl-N3-(2,3-dihydro-1H-inden-2-yl)-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}azepane-4-carboxamide
2-({[2-(diethylamino)ethyl]amino}methyl)-6-methylquinolin-4-ol
N-(2-acetamidophenyl)-2-{methyl[2-(oxan-2-yl)ethyl]amino}acetamide
(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
N4-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-6-methylpyrimidine-2,4-diamine
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
N-ethyl-N-methyl-2-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
methyl N-(1-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-1-oxopropan-2-yl)carbamate
1-[3-(3-methoxypropyl)piperidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
1-(2-aminoethyl)-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{[5-(3-chlorophenyl)furan-2-yl]methyl}-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
2-[(5-methylpyrazin-2-yl)methyl]-9-(morpholine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(3-methoxyphenoxy)ethyl]pyridine-4-carbonitrile
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
2-{4-[4-(morpholin-4-yl)butyl]-1,4-diazepan-1-yl}-1,3-benzothiazole