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N-methyl-3-(2-oxo-1,2-dihydropyridin-1-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
methyl 4-(4-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)benzoate
1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-4-(piperidin-1-yl)butan-1-one
1-(5-methanesulfonyl-2-methylphenyl)-3-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-{2-[3-(propan-2-yloxy)phenyl]ethyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
6-chloro-3-fluoro-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
6-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
3-(2,5-dioxoimidazolidin-4-yl)-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methylpropanamide
2-[9-(cyclopentylcarbamoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
8-(4-aminopyrimidin-2-yl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]-3-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]urea
1-{4-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]phenyl}ethan-1-one
(3S,4S)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
N-(1-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
N-butyl-N-methyl-3-(pyrrolidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[(3-methylphenyl)methyl]-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazine
3-[3-(dimethylamino)propyl]-8-{[3-(methylsulfanyl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(propan-2-yl)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidin-4-amine
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl)(quinolin-8-ylmethyl)amine
1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-amine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}piperidin-2-one
3-(2-oxoazepan-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
methyl 6-(butan-2-yl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[(2-{1-cyclohexyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]-1H-pyrazole
7-(pyridin-3-yl)-4-(1,3-thiazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-(1-benzofuran-2-ylmethyl)-6-oxa-9-azaspiro[4.5]decane
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl][(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1-(oxan-4-yl)piperidine-4-carboxamide
1-[(4-methyl-1H-imidazol-5-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
methyl 2-oxo-3-(pentan-3-yl)-1-(1,3-thiazol-5-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
2-{1-[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-2-methoxyethyl}pyridine
4-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
N-[(2-chlorophenyl)methyl]-3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[2-(propylsulfanyl)phenyl]piperazine-1-carboxamide
2-[7-(2,2-dimethylpropyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
5-[1-(furan-2-ylmethyl)pyrrolidin-2-yl]-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]thiophene-2-carboxamide
4-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carbonyl}thiomorpholine
3-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-methyl-5-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}pyrimidin-2-amine
2-(2-hydroxyethyl)-8-[3-(3-methoxyphenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(phenylsulfanyl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyrrolidine-1-carbonyl)piperazine
2-[4-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)phenyl]-3,4,5,6,7,8-hexahydroquinazolin-4-one