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2-(1H-imidazol-1-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)acetamide
6-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
2-benzyl-4-(3-chlorobenzoyl)morpholine
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
5-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-(3-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)-2,3-dihydro-1H-isoindol-1-one
2-methoxy-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyridine-3-carboxamide
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}benzamide
2-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
4-(2-ethoxyethyl)-N-[2-(prop-2-en-1-yloxy)phenyl]piperazine-1-carboxamide
1-(2-methylpropanoyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
[(1-cyclopentylpiperidin-4-yl)methyl]({[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl})(pyridin-3-ylmethyl)amine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2-phenoxyethyl)piperidine
3-[(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)methyl]benzoic acid
N-[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[(2-ethoxyphenyl)methyl]cyclopropanamine
3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyrazin-2-yl)ethyl]pyridin-2-amine
(4aS,7aR)-1-(4-fluorobenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(3-oxo-3-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propyl)piperidin-2-one
(2R,3S,6R)-5-(2,6-dimethylpyridin-4-yl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
{7-[6-(azepan-1-yl)pyridazin-3-yl]-5-chloro-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-ethyl-1-[1-(1-phenylethyl)-1H-pyrazol-5-yl]-3-(propan-2-yl)urea
[1-(5-fluoro-2-methylbenzenesulfonyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
2-(2H-1,3-benzodioxol-5-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
4-(2-{1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]piperidin-2-yl}ethyl)phenol
1-(2-fluoro-5-methanesulfonamidophenyl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
2-cyclohexyl-N-[(3-methoxyphenyl)methyl]-N-methyl-1,3-benzoxazole-6-carboxamide
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
6-methyl-1-(3-oxo-3-{spiro[indene-1,4'-piperidine]-1'-yl}propyl)-1,2-dihydropyridin-2-one
(3R,5S)-N-[2-(1H-indol-3-yl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-phenylazepane
[2-(1,3-benzoxazol-2-yl)phenyl]methanol
N-(2-methoxyphenyl)-3-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propanamide
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](methyl)({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
3,5,7-trimethyl-2-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-indole
2-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}pyridine
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-[(2-fluorophenyl)methyl]piperidin-2-one
3-(4-tert-butylbenzoyl)-1-(oxane-4-carbonyl)piperidine
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
8-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)ethan-1-one
4-(1-propyl-1H-imidazol-2-yl)-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(furan-2-ylmethyl)-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanamide
2-(2-{[4-(morpholin-4-yl)piperidin-1-yl]methyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
ethyl 1-{1-[2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperidin-4-yl}piperidine-3-carboxylate
3-[(dimethylamino)methyl]-1-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)pyrrolidin-3-ol
1'-(3-chloropyridin-2-yl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]