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1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-2-(3-methoxyphenyl)piperidine
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(5-fluoro-2-methoxyphenyl)-2-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}acetic acid
(1R,2S,6R,7S)-4-{[3-(morpholin-4-yl)phenyl]methyl}-4-azatricyclo[5.2.2.02,6]undecane
3-{[(3-methyloxetan-3-yl)methyl]sulfamoyl}-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
methyl 3-methyl-4-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}amino)benzoate
1-(5-fluoro-1H-indole-2-carbonyl)-4-propyl-1,4-diazepan-5-one
1-{3-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
N-[(3-hydroxypyrrolidin-3-yl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,4S)-1-(butane-1-sulfonyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(3-methoxyphenyl)methyl]acetamide
6-{[benzyl(methyl)amino]methyl}-N-[(4-chlorophenyl)(phenyl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
6-(2,5-dimethylphenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-ethyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)-N-(oxan-4-ylmethyl)acetamide
1-[1-(6-chloroquinolin-2-yl)piperidin-4-yl]-3-methylbutan-1-ol
1-cyclopentyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyrimidine
N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}oxolane-3-carboxamide
5-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]pyrazin-2-ol
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
7-[(3,4-difluorophenyl)methyl]-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-2-(pyridin-3-yl)acetamide
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}imidazolidine-2,4-dione
3-[(2-chloro-4-fluorophenyl)methyl]-5-(3-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazole
3-methoxy-5-{[3-(methylsulfanyl)propyl]carbamoyl}benzoic acid
2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
(4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-1,4-oxazepan-6-yl)methanol
1-cyclopentyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-6-oxopiperidine-3-carboxamide
N-(4-fluoro-2-methylphenyl)-2-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}acetamide
N-[1-(4-chlorophenyl)cyclobutyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
1-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
1-[4-(2,5-dimethoxybenzoyl)benzoyl]-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
N-(5-methyl-2,1,3-benzothiadiazol-4-yl)-4-(3-methylpyridin-2-yl)piperazine-1-carboxamide
4-{[2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
4-{1-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-2-yl}phenol
N,2-dimethyl-N-(1-{1-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]piperidin-4-yl}-2-phenylethyl)furan-3-carboxamide
5-{[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}-2,1,3-benzoxadiazole
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[(5-fluoro-1H-indol-2-yl)methyl]methylamine
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-[3-(3-methylphenyl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
N-methyl-2-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]-N-(propan-2-yl)acetamide
4-(hydroxymethyl)-1-[4-(4-methylpiperazin-1-yl)benzoyl]azepan-4-ol
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
(1S,5R)-6-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-(trifluoromethyl)benzamide
3-{5-[2-(oxolan-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[1-(pyridin-3-yl)propyl]quinoline-4-carboxamide
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine