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(3R,4R)-1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-4-ethylpiperidine-3,4-diol
(3R,5R)-N-benzyl-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carboxamide
1-methyl-5-(thiomorpholin-4-yl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-methyl-2-[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
N-[2-(3-fluorophenyl)ethyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methylpiperidine-3-carboxamide
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-5,5-diphenylpiperidin-2-one
7-methyl-4-{2-oxo-2-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethyl}-2H-chromen-2-one
7-(5-chloropyridine-2-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(benzylsulfanyl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
(3S,4S)-1-(morpholine-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-chloro-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-(piperidin-1-yl)benzamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
3-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-ethyl-3-methyl-8-(quinolin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(6-cyanopyridin-3-yl)phenyl]acetamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-2-phenoxyethan-1-one
4-(4-methoxybenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1'-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N4-(3-phenoxypropyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(quinoxaline-2-carbonyl)piperazin-2-one
2-ethoxy-5-(2-phenylpyrimidin-4-yl)benzoic acid
2-(4-benzylmorpholin-2-yl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
N-(oxan-4-ylmethyl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
5,6-dimethoxy-2-(pyrrolidin-3-ylmethyl)-1,2-dihydroisoquinolin-1-one
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-(oxane-2-carbonyl)piperidine
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
4-(4-methanesulfonylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
8-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazole-3-carbonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-[3-(4-methanesulfonylphenyl)phenyl]-1-(2-methylprop-2-en-1-yl)-1H-pyrazole
1-[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(3aS,6aS)-5-(5-chloropyridin-2-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S)-2-amino-1-[2-(dimethylamino)-4-(4-hydroxypiperidin-1-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-3-hydroxypropan-1-one
6-{2-methylthieno[3,2-d]pyrimidin-4-yl}-5,6,7,8-tetrahydro-1,6-naphthyridine
4-cyclobutyl-6-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}pyrimidin-2-amine
7-(1,3-benzothiazol-2-yl)-4-[(2,5-difluorophenyl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclopropyl-5-(2,6-dimethylpyrimidine-4-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
[(3R,4S)-1-[(2,3-dichlorophenyl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-[2-(4-methoxyphenyl)ethyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
N-methyl-5-propyl-N-(quinoxalin-6-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(3,3-diphenylpiperidin-1-yl)-N-methylpyridine-4-carboxamide
5-{2-[(4aS,8aR)-2-oxo-1-propyl-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N3-[2-(3,4-dimethoxyphenyl)ethyl]-N3-methyl-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(quinolin-2-ylmethyl)piperidin-4-yl]oxy}benzamide