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N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-methylazepane-2-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}pyridine-3-carboxamide
N-[3-(methylsulfanyl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
3-{[2-(1-cyclohexyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl](methyl)amino}-1λ6-thiolane-1,1-dione
(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazol-4-yl)methanol
4-{3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]benzoyl}morpholine
2-(4-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
3-methoxy-1-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,2-dihydropyridin-2-one
N-(2,3-dihydro-1H-inden-2-yl)-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylfuran-2-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]thiophene-3-carboxamide
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2,2-dimethylmorpholine
4-[(diethylamino)methyl]-5-ethyl-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}furan-2-carboxamide
5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)-5-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
(3aR,7aS)-2-(1-benzylpyrrolidine-2-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(2S,4R)-4-amino-1-(2,3-dihydro-1H-indene-5-carbonyl)-N-methylpyrrolidine-2-carboxamide
2-[(3S,4R)-3-methanesulfonamido-4-(propan-2-yl)pyrrolidin-1-yl]-N-(2-phenylethyl)acetamide
1-ethyl-3-(propan-2-yl)-5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
7-fluoro-2-methyl-4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]quinoline
2-phenyl-7-[3-(pyridin-3-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[(3-methyloxetan-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-{1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
5-fluoro-3-methyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
3-[2-(4-fluorophenyl)ethyl]-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
1-[(2,2-dimethyloxan-4-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
8-[(4-hydroxyphenyl)methyl]-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(3-chloropyridin-2-yl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N,N-dimethyl-5-({methyl[3-(pyrrolidin-1-yl)propyl]amino}methyl)pyridin-2-amine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(dimethyl-1,3-thiazole-5-carbonyl)piperidine
(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)(thiophen-2-ylmethyl)amine
1-ethyl-N-methyl-5-[methyl(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-benzyl-1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-ethyl-1,4-diazepan-5-one
2-{1-[2-(4-fluorophenoxy)ethyl]piperidin-4-yl}propan-2-ol
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
3-({[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylpropanamide
2-[(1-benzyl-1H-imidazol-5-yl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2-fluorobenzenesulfonyl)piperidine
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(3-chloro-4-fluorophenyl)-3-[1-(furan-2-carbonyl)piperidin-4-yl]propanamide
7-methoxy-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(2-ethoxyphenyl)-3-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]urea
(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
5-fluoro-2-[1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
2-tert-butyl-5-[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
9-(2-amino-6-methoxypyrimidin-4-yl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methoxyphenyl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one