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(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(4-fluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[2-(4-cyclopropanecarbonyl-1,4-diazepan-1-yl)-2-oxoethyl]-1,2-dihydroquinolin-2-one
2-ethyl-9-[(3-fluoro-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(but-2-yn-1-yl)-1-[(1-ethylpyrrolidin-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-methyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(2-phenylethyl)piperidin-3-amine
methyl 4-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)benzoate
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,3,5-trimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
(benzylsulfamoyl)(ethyl)(pyridin-4-ylmethyl)amine
2-(2,3-dihydro-1H-inden-1-yl)-N,N-bis(2-hydroxyethyl)acetamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
4-{[2-(methoxymethyl)piperidin-1-yl]methyl}benzoic acid
(1R,3S)-7-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-7-azaspiro[3.5]nonane-1,3-diol
4-(3-ethoxyphenyl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
1-{3-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]phenyl}ethan-1-one
(4aS,7aR)-1-[(4-ethylphenyl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2H-1,3-benzodioxol-5-yl)-1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
N-{[8-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}cyclopentanamine
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-6-(propan-2-yl)pyrimidin-4-amine
N-[(2-chloro-6-fluorophenyl)methyl]-2-(trifluoromethyl)pyrimidin-4-amine
N-[3-(1H-indazol-1-yl)propyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine-4-carboxylic acid
3-[(3S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)piperidin-3-yl]-1-[4-(2-methoxyphenyl)piperazin-1-yl]propan-1-one
4-{[(2S,4S)-4-amino-2-[(propan-2-yl)carbamoyl]pyrrolidin-1-yl]sulfonyl}benzoic acid
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline-4-carboxylic acid
N-[1-(2-phenylethyl)piperidin-3-yl]-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
1-(2,6-dimethylpyridin-4-yl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
3-(2H-1,3-benzodioxol-5-yl)-1-[4-(methoxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
N-[(5-methylfuran-2-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-4-oxo-4-phenylbutanamide
1-(cyclopropylmethyl)-5-(isoquinoline-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-cyclopentyl-2-{[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]amino}propanamide
(3R,4S)-1-(4,6-dimethylpyrimidin-2-yl)-4-propylpyrrolidin-3-amine
2-(3-chlorophenyl)-2-hydroxy-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
3-(4-cyano-2-fluorophenyl)-1-(oxan-4-ylmethyl)urea
(3S,4R)-1-(4-chloro-3-fluorobenzoyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[4-({methyl[1-(3-phenylpropyl)piperidin-3-yl]amino}methyl)phenyl]acetamide
N-(2-methoxyethyl)-2-[2-(1H-pyrazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
N-(oxolan-2-ylmethyl)-3-[(pyrimidin-4-ylmethyl)sulfamoyl]benzamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
4-{[1-(2-chlorobenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
[(3-{[1-(benzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
1,3-dimethyl-6-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-(quinoxalin-2-yl)pyrrolidin-3-yl]methanol
1-cyclopropyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
3-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methylurea
2-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
1-(1H-imidazol-2-ylmethyl)-3-(6-methoxynaphthalene-2-carbonyl)piperidine
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(3-methoxypropyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(5-methyl-1,3-thiazol-2-yl)-3-({methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)benzamide