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N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-hydroxy-3-methylbutanamide
2-{4-[(2-chlorophenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-{2-methyl-1-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]propan-2-yl}morpholine
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-[1,3-dioxo-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]piperidine-4-carboxamide
2-[5-(4-chloro-2-fluorophenyl)-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
2-methyl-6-(1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)pyrimidin-4-ol
2-methyl-8-[6-(morpholin-4-yl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane
1-{[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
2-phenoxy-1-[3-(pyridin-2-yl)azetidin-1-yl]butan-1-one
8-(dimethyl-1,3-oxazole-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-4-(quinolin-4-ylmethyl)piperazine-2-carboxamide
3-(1H-pyrazol-1-ylmethyl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-(1-methyl-1H-pyrrol-3-yl)acetamide
methyl({phenyl[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
(1S,5R)-3-benzoyl-6-(1-methyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
5-(1H-imidazol-1-ylmethyl)-2-[3-(2-methylphenyl)piperidin-1-yl]pyridine
2-(furan-2-yl)-7-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{[1-tert-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-methyl-1H-1,3-benzodiazole
2-(1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazol-2-yl}-N-methylformamido)-N-methylacetamide
5-[(4-ethyl-3,3-dimethylpiperazin-1-yl)methyl]-2-methoxypyrimidine
N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N-(pyridin-2-ylmethyl)acetamide
1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-8-(thiophen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
{1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
2-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
7-(1,3-benzothiazol-2-yl)-4-[(4-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-(morpholine-4-carbonyl)phenyl]-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]piperidin-4-amine
2-cyclooctyl-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
5-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-2-(propylsulfanyl)pyrimidine
3-(1H-indol-3-yl)-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}propanamide
4-[(2-fluorophenyl)methyl]-1-(3-phenylpropyl)-1,4-diazepan-5-one
2-methoxy-6-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
4-[(3-chlorophenyl)methyl]-1-(furan-2-ylmethyl)-1,4-diazepan-5-one
(3R,4R)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
(3aS,6aR)-5-[(2,4-difluorophenyl)methyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-cyclopropyl-N-ethyl-N-(2-hydroxyethyl)-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
1-(6-chloro-2-methylpyridin-3-yl)-3-[2-(ethanesulfonyl)ethyl]urea
N-cyclopropyl-2-ethyl-7-(oxane-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2-aminopyridin-3-yl)methyl]-2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
8-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-butylphenyl)urea
2-(1,2-benzoxazol-3-yl)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]acetamide
1-[2-({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
2-[(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)amino]propan-1-ol