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2-{3-[(3,4-dimethylpiperazin-1-yl)methyl]phenoxy}acetamide
5-acetyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}thiophene-2-carboxamide
1-{4-[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amino]piperidin-1-yl}ethan-1-one
3-methoxy-N-(3-oxo-3-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}propyl)benzamide
8-cyclopropyl-9-oxo-N-[2-(thiophen-2-yl)ethyl]-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-[5-(3-acetylphenyl)-1H-indazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
5-ethyl-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3,4-oxadiazol-2-amine
4-[(4-methyl-5-{1-[(5-methylpyrazin-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
1-[(1-ethylpyrrolidin-2-yl)methyl]-3-(oxan-2-ylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-{3-oxo-3-[4-(2-phenoxyethyl)piperazin-1-yl]propyl}piperidin-2-one
1-ethyl-4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine
7-(4-chlorophenyl)-2-[(ethylsulfanyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
9-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)piperazine-2-carboxylic acid
3-methyl-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1,2-dihydroquinoxalin-2-one
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-imidazol-1-yl)propan-1-one
5-(dimethylamino)-2-{2-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
(2R)-2-amino-4-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pentanamide
4-(2,3-dimethylphenyl)-6-methoxypyrimidin-2-amine
[(3R,4R)-1-(5-chloro-2-methoxybenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-(3-methoxybenzoyl)-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-methyl-1,4-diazepan-5-one
3-{benzyl[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}-2-methylpropan-1-ol
5-(3-methoxyphenyl)-3-[2-(pyridin-2-yl)pyrrolidin-1-yl]-1,2,4-triazine
(4S)-3-[2-(2,3-dimethylphenoxy)ethyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
2-ethyl-8-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
8-(but-3-en-1-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-2-phenylethan-1-one
1-(4-{[(3-fluorophenyl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[2-(4-chlorophenyl)ethyl]-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
6-ethyl-4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methylquinoline
2-(2-methoxyphenoxy)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
(3aR,7aS)-2-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
2-chloro-N-[2-(pyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
2-(3-phenylpiperazin-1-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(pyridin-3-ylmethyl)-1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-(1-{7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
1'-(3-fluoro-4-methylbenzoyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3aR,6aR)-2-(5-acetylpyridin-2-yl)-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(azepan-1-ylmethyl)-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
1'-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}oxolane-2-carboxamide
6-{2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carboxylic acid
5-(dimethyl-1,3-thiazol-5-yl)-8-methoxyquinoline
methyl 3-[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]propanoate
4-[2-(2-phenylethyl)piperidin-1-yl]butan-1-ol