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3-(2-ethyl-1H-imidazol-1-yl)-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}propanamide
N-benzyl-5-(4H-1,2,4-triazol-4-yl)pyridin-2-amine
1-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}-2-methyl-1,4-diazepan-5-one
4-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
2-(isoquinolin-5-yl)benzamide
2-(5-chlorothiophene-2-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
4-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-1,4-oxazepane
N,N-diethyl-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
(2R)-2-(methoxymethyl)-1-(5-methyl-2-phenylfuran-3-carbonyl)pyrrolidine
N-[(5-{[6-(dimethylamino)pyridin-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]methanesulfonamide
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-4-phenylpyrimidin-2-amine
4-(4,4-difluoropiperidine-1-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
5-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,1,3-benzothiadiazole
8-[(3-fluoro-2-methylphenyl)methyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]propanamide
1,9-dimethyl-4-{thieno[3,2-d]pyrimidin-4-yl}-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-ethyl-3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]urea
(3R,4R)-1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
2-(dimethyl-1,2-oxazol-4-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
(1R,5R)-6-(cyclobutylmethyl)-3-(dimethyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-methyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-methyl-8-[2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-(5-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
1-(3-methoxyphenoxy)-3-[(thian-4-yl)amino]propan-2-ol
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[(4-methyl-1,3-thiazol-2-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
(1-{[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)(phenyl)methanol
(1S,5R)-6-benzyl-3-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(4S,6R)-N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
6-amino-N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]pyridine-3-carboxamide
2-(3-methoxypropyl)-8-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-(benzyloxy)-1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
2-methyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]-1,4-diazepan-5-one
4-(4-chlorophenyl)-1-[2-(2-methoxyphenoxy)ethyl]piperidin-4-ol
(1R,5R)-6-benzyl-3-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[(dipropylamino)methyl]benzamide
2-(3-chloro-1-benzothiophen-2-yl)-1-(2-methanesulfonylethyl)-1H-imidazole
2-fluoro-6-hydroxy-N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]benzamide
(3aR,6aR)-2-[(4-fluoro-3-methoxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-4-{4-[7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}but-3-yn-2-ol
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
ethyl 1-(3-chlorophenyl)-5-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole-4-carboxylate
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-1,2,5-thiadiazole-3-carboxamide
N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-(pyrimidin-4-yl)piperidine-1-carboxamide