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2-{1-[(2R)-oxolane-2-carbonyl]pyrrolidin-2-yl}-1,3-benzothiazole
N-[(2-fluorophenyl)methyl]-3-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propanamide
4-[4-(furan-2-yl)benzoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
2,2-dimethyl-N-[3-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)pyridin-2-yl]propanamide
N-[(1-ethylpiperidin-4-yl)methyl]-1-benzofuran-2-sulfonamide
1-({5-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)-4-methylpiperazine
5-(2,6-dimethylphenoxymethyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1,2-oxazole-3-carboxamide
5,6-dimethyl-2-[4-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
1-(azocan-1-yl)-3-(2-methoxy-5-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenoxy)propan-2-ol
1-[(3-fluoro-4-methylphenyl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
1'-[(5-cyclopentylthiophen-2-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-propylurea
2-[3-(furan-2-yl)-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
[2-({4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-(4-tert-butyl-1,3-thiazol-2-yl)-2-{[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}acetamide
3-phenoxy-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-(1H-imidazol-1-yl)acetamide
3-(2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)pyridine
N-[2-(3-chlorophenoxy)ethyl]-N-ethyl-1,3-dimethyl-1H-pyrazole-5-carboxamide
9-{[2-(prop-2-yn-1-yloxy)phenyl]methyl}-3-oxa-9-azaspiro[5.5]undecane
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,2,5-trimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
methyl 3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]benzoate
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
3-{2-[2-(3-fluorophenyl)azepan-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
2-[methyl(2-phenylethyl)amino]-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
5-{6-amino-5-cyano-4-[3-(2-hydroxyethoxy)phenyl]pyridin-2-yl}thiophene-3-carboxylic acid
2-(2,5-dimethylphenoxy)-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]propanamide
methyl 1-(2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetyl)piperidine-4-carboxylate
(1R,7S)-N-(1H-imidazol-2-ylmethyl)-N-methyl-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[5-(ethylcarbamoyl)-2-methylphenyl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
5-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[3-(1H-pyrazol-1-yl)propyl]propanamide
2-(4-{[3-(aminomethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
2-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]propane-1,3-diol
1-[1-(1-benzofuran-5-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
4-{5-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-3,5-dimethyl-1,2-oxazole
6-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
4-chloro-5-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-ethyl-4-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)pyrimidine
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
methyl 4-{[methyl({[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}benzoate
4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2,6-dimethoxyphenol
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(3-hydroxypropyl)piperidine-4-carboxamide
3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
2-(5-methyl-2-oxo-5-phenylpiperidin-1-yl)acetic acid
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(furan-2-yl)-N-methylbenzamide
1-butyl-5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)pyrrolidin-2-one
2-[(2-{[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]carbamoyl}phenyl)amino]acetic acid
N-(cyclohex-1-en-1-ylmethyl)-1-methylazepane-2-carboxamide