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2-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzoic acid
N-(5-chloro-2-methoxyphenyl)-3-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]propanamide
N-{[1-(3-fluorophenyl)cyclopentyl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[2-(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-4-methoxybenzamide
3-{3-methyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxymethyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
5-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
(1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperidin-3-yl)methanamine
3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-(difluoromethyl)-1H-pyrazole
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-(4-methylphenyl)quinoline-4-carboxamide
methyl 6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-3-[2-(2-methylphenyl)acetamido]thieno[2,3-b]pyridine-2-carboxylate
1-benzyl-4-[(2-fluoro-4-methoxyphenyl)methyl]-6-methoxy-1,4-diazepan-2-one
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-methylbutanamide
2-(naphthalen-2-yl)-5-[(4-propylpiperazin-1-yl)methyl]pyrimidine
3-[1-(5-acetylthiophene-3-carbonyl)piperidin-4-yl]-N-phenylpropanamide
1-[1-(2-amino-9H-purin-6-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]acetamide
1-(1,2-oxazole-5-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
N-propyl-4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
(3S,4S)-1-[2-(methylamino)pyrimidine-5-carbonyl]-4-propylpyrrolidine-3-carboxylic acid
N-[4-({4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenyl]acetamide
1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-phenylpiperidine
3-methyl-7-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
{5-fluoro-7-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
5-(morpholin-4-ylmethyl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}furan-3-carboxamide
(1S,6R)-9-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-methanesulfonyl-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]-1H-1,3-benzodiazole
3-cyclohexyl-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1H-pyrazole-4-carboxamide
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](quinolin-3-ylmethyl)amine
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-4-phenoxybutan-1-one
2-(methylamino)-N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
2-(1-acetylpiperidin-4-yl)-7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidine
3-{2-[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}-5-ethyl-1,2,4-oxadiazole
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-propylpyridine-4-carboxamide
8-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(2E)-1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-3-(thiophen-2-yl)prop-2-en-1-one
2,6-dimethyl-4-({[2-(pyridin-4-ylformamido)ethyl]amino}methyl)phenyl acetate
N-(2-{[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)acetamide
1-(2-cyclopropylacetyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-(pyridin-4-ylmethyl)-9-[(1r,4r)-4-methylcyclohexanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
ethyl 4-{1-ethyl-3-methyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}piperidine-1-carboxylate
1-(2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydroquinolin-2-one
[(6-chloropyridin-3-yl)methyl]({4-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)amine
[2-(1H-imidazol-1-yl)ethyl](methyl){[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
1-{2-hydroxy-3-[3-(1,2-oxazolidin-2-ylmethyl)phenoxy]propyl}piperidin-4-ol
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-[5-(propan-2-yl)pyrimidin-2-yl]piperidin-3-yl]methanol