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N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(prop-2-en-1-yloxy)benzamide
1-[(4-fluoro-3-methoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
7-(cyclopropylmethyl)-2-[4-(dimethylamino)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
2-(azepan-1-yl)-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
2-{1-[(5-methylfuran-2-yl)methyl]-4-[(2E)-4-methylpent-2-en-1-yl]piperazin-2-yl}ethan-1-ol
6-[(4-chlorophenyl)amino]-1-[2-(1H-pyrrol-1-yl)ethyl]-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
2-(1H-indol-1-yl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
4-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]ethyl}morpholine
2-{[5-(2-methyl-1,3-oxazol-4-yl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-{[4-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-1-yl]methyl}phenol
5-methoxy-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
4-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
dimethyl(3-{2-[1-(naphthalene-1-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
4-({2-[1-(benzenesulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
6-amino-N-[(3R,5S)-5-(ethylcarbamoyl)-1-(furan-2-carbonyl)pyrrolidin-3-yl]pyridine-3-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
4-(4-fluorophenyl)-N-[(3-methyloxetan-3-yl)methyl]-4-oxobutanamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
4-{[4-(diphenylmethyl)piperazin-1-yl]methyl}pyrimidine
1-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-6-(pyridine-3-sulfonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-{[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}-1-methyl-1,2-dihydropyridin-2-one
6-({[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}amino)pyrazine-2-carboxamide
N-(2,2-diphenylethyl)-2-(morpholin-3-yl)acetamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]propanamide
3-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1-{3-[(pyridin-3-yl)amino]propyl}urea
7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[5-(2,1,3-benzoxadiazol-4-ylmethyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
2-{[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}-1-(pyridin-3-yl)ethan-1-ol
5-[3-(1H-pyrazol-1-yl)propyl]-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
N-(1-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-cyclopentyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-5-oxopyrrolidine-3-carboxamide
2-[5-(3-chloro-5-fluoro-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethan-1-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-indazole-3-carboxamide
7-methoxy-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[2-(pyridin-2-yl)ethyl]-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-N-(propan-2-yl)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidine-2-carboxamide
(1S,5R)-6-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(pyridin-4-ylmethyl)propanamide
4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1,4-oxazepan-6-ol
1-cyclopentyl-4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyrrolidin-2-one
N-[(5-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
3-[6-hydroxy-4-(2-phenylacetyl)-1,4-diazepan-1-yl]pyrazine-2-carbonitrile
4-(2,6-dimethylquinoline-4-carbonyl)-3-(2-hydroxyethyl)piperazin-2-one