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methyl 5-(cyclopentylamino)-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-ethyl-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(morpholin-4-yl)pyrimidin-4-amine
3-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1H-pyrazol-5-amine
N-(dimethyl-1,2-oxazol-4-yl)-3-{[ethyl(oxolan-2-ylmethyl)amino]methyl}benzamide
4-(1H-imidazol-1-yl)-N-(oxolan-2-ylmethyl)-N-{[4-(pyridin-3-ylmethoxy)phenyl]methyl}benzamide
4,4-difluoro-1-[4-(piperidin-3-yl)benzoyl]piperidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(4aS,7aR)-1-(1-aminocyclopropanecarbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-2-({1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-({4-[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]piperazin-1-yl}methyl)benzonitrile
3-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine
1-(2-methoxyethyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-methoxyacetamide
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]acetamide
4-[(5-ethylpyridin-2-yl)methyl]-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
2-methoxy-2-methyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-3-(3-chloro-1,2-oxazol-5-yl)propan-1-one
2-[1-(2H-1,3-benzodioxol-5-yl)-5-[(dimethyl-1,3-thiazol-5-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
3-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1,3-dimethyl-2,6-dioxo-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
6-methyl-4-oxo-2-(2-phenylethyl)-N-(propan-2-yl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
7-methoxy-3-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,3,4,5-tetrahydro-1H-3-benzazepine
3-{[(2-chlorophenyl)formamido]methyl}-N-(2-phenylethyl)piperidine-1-carboxamide
1-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-{6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-3-carbonyl}morpholine
N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
5-{4-[(4-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
5-[3-({[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}methyl)pyrrolidin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
{1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)phenyl]ethyl}dimethylamine
1-methyl-3-{2-[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]-1H-imidazol-1-yl}pyrrolidin-2-one
2-(2,3-dimethoxy-5-methylphenyl)-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
N-[phenyl(pyridin-4-yl)methyl]-5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-(3-hydroxy-3-phenylpropyl)-1-methyl-3-(2,4,6-trimethylpyridin-3-yl)urea
2-amino-4-(2-chloro-4-hydroxyphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-ethylpiperidin-3-ol
(4aS,8aR)-6-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
(3aR,6aR)-2-cyclopentyl-N-[2-(1H-imidazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[2-(dimethylamino)ethyl]-N-[(4,6-dimethylpyridin-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-(1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-[(oxolan-3-yl)sulfamoyl]-N-(2-phenylethyl)benzamide
1-(2-methoxybenzoyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazine
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
2-(2-methylphenyl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine
5-(2-fluorophenyl)-N-[1-(pyrazin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
[3-benzyl-1-(2-methyl-1-phenyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-3-yl]methanol
N-[(2S,4R,6S)-2-benzyl-6-(5-tert-butyl-1H-pyrazol-3-yl)oxan-4-yl]acetamide