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(3S,5R)-N3-(4-methylphenyl)-N5-{[4-(methylsulfanyl)phenyl]methyl}piperidine-3,5-dicarboxamide
6-(2-aminoethyl)-N-[1-(3,5-difluorophenyl)ethyl]pyrimidin-4-amine
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(2S,4R)-N-ethyl-1-(1H-imidazol-4-ylmethyl)-4-[3-(4-methyl-1H-pyrazol-1-yl)propanamido]pyrrolidine-2-carboxamide
3-[(3-chlorophenyl)methyl]-1-(2,6-diaminopyrimidin-4-yl)piperidine-3-carboxylic acid
(3S,4S)-4-(naphthalen-2-yl)-1-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-3-ol
2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]cyclobutanecarboxamide
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
3-(1,2-oxazinan-2-yl)-N-(thiophen-2-ylmethyl)propanamide
N-[(3S,4R)-1-[(2-methoxyphenyl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylphenyl)piperazin-2-one
N-ethyl-2-[4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-1-yl]acetamide
1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(2-methylpropyl)piperidine-3-carboxamide
N-(pyridin-2-ylmethyl)-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
6-(5-fluoro-2-methoxybenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-[methyl(pyridin-3-ylmethyl)amino]-N-[2-(2-methyl-1H-indol-3-yl)ethyl]acetamide
2-methoxy-5-{1-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazol-2-yl}pyrimidine
N-(2H-1,3-benzodioxol-5-yl)-1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-amine
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N,6-dimethyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N,1-dimethylpiperidin-4-amine
2-{[5-(4-cyanophenyl)-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-(dimethylamino)-2-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}propanamide
4-ethyl-1-methyl-3-{[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 5-[2-(prop-2-en-1-ylsulfanyl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-({5-[(2-chloro-3,6-difluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-[(5-cyclohexylthiophen-2-yl)methyl]-3-methoxypyrrolidine
1-(2-methoxyphenyl)-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperazin-2-one
2-{2-[(3-hydroxy-3-methylbutyl)(methyl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
ethyl 1-[1-(1H-imidazol-1-yl)butan-2-yl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
2-(4-methoxyphenoxy)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
3-(1,1-dioxo-1λ6-thiolan-3-yl)-1-[3-(3-methoxyphenyl)phenyl]-3-methylurea
1-(7-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3,3-dimethylbutan-1-one
3-{1-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}phenol
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}piperazine-2-carboxylic acid
3-benzyl-5-[2-(thiophen-2-yl)ethyl]-1H-1,2,4-triazole
N-[(2-ethoxyphenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)-1,6-dihydropyridine-2-carboxamide
(2R,3R)-1'-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(piperidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(dimethylamino)-1-[3-(2-fluorophenoxy)azetidin-1-yl]-2-(4-fluorophenyl)ethan-1-one
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-(thiophen-2-yl)pyrimidine
2-methoxy-3-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridine
(1R,5R)-6-(cyclobutylmethyl)-3-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,2,3,4-tetrahydroisoquinoline
8-{[2-(furan-2-yl)phenyl]methyl}-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-6-methyl-4H-pyran-4-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
5-{4-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
1'-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2,3-dimethylquinoxaline-6-carboxamide