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(1-{[1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
2-({2-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methylpyridine
1-(2-methoxyethyl)-4-({2-[2-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}methyl)pyrrolidin-2-one
5-benzyl-1-(3-methoxyphenyl)-4-(2-methylpropanoyl)piperazin-2-one
2-chloro-5-(1-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
1-(3-chloro-4-methoxyphenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-methyl-5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]pyrimidine
N-cyclopentyl-1-[1-(furan-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
8-methoxy-2-methyl-5-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}quinoline
(2S,4R)-4-(dimethylamino)-1-{[2-(propylamino)pyrimidin-5-yl]methyl}pyrrolidine-2-carboxylic acid
N-methyl-4-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}benzene-1-sulfonamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
5-{1-[2-(2-butyl-5-chloro-1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}-3-ethyl-1,2,4-oxadiazole
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methylpropan-1-one
3-[(3R,4S)-1-(3-ethoxybenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-(4-{[(4-methoxyphenyl)methyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
2-[3-({[(3S)-1-benzylpyrrolidin-3-yl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
(4S)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
[(1-ethyl-1H-pyrazol-4-yl)methyl]({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-(2-chlorophenoxy)-1-(thiophene-2-carbonyl)azetidine
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[4-(hydroxymethyl)phenyl]methyl}acetamide
1-benzyl-4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
N-methyl-3-{3-methyl-3,9-diazaspiro[5.6]dodecane-9-carbonyl}pyridin-2-amine
4-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}thiomorpholine
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-5-methylpiperidin-2-one
9-[2-(propylsulfanyl)acetyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-[2-(4-methyl-1,4-diazepan-1-yl)acetamido]cyclobutane-1-carboxylate
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-methoxy-1-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2,3,4-trifluorobenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(2R)-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-phenylpropan-1-one
2-(3-phenylpiperidine-1-carbonyl)-1H-1,3-benzodiazole
3-[1-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
1-benzyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(2S)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]pyrrolidine-2-carbonyl]morpholine
3-[5-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl](methyl)amino}methyl)thiophen-2-yl]prop-2-yn-1-ol
6-[({[5-(2-chlorophenyl)furan-2-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
2-[({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)(methyl)amino]-N-methylacetamide
7-(3-methoxyphenyl)-2-(5-methyl-1,2-oxazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylate
N-{[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-3-yl]methyl}-4-fluorobenzamide
2-fluoro-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-sulfamoylbenzamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
4'-[(2-methyl-1,3-oxazol-4-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 3-[(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)carbamoyl]propanoate
1-(4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}thiophen-2-yl)ethan-1-one